SCHEMBL6949095

SCHEMBL6949095

CCOc1ccc2cc(CCCC(=O)N3CCCC(Cc4ccccc4)C3)[nH]c2c1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 3/20 0.47
KMT2A Q03164 3/20 0.47
NPC1 O15118 1/20 0.47
ALDH1A1 P00352 5/20 0.42
KDM4E B2RXH2 3/20 0.42
MAPK1 P28482 2/20 0.42
HPGD P15428 3/20 0.41
TSHR P16473 1/20 0.41
HSD17B10 Q99714 1/20 0.41
SMN1; SMN2 Q16637 1/20 0.41
TACR3 P29371 1/20 0.40
CYP1A2 P05177 1/20 0.40
CYP3A4 P08684 1/20 0.40
CYP2D6 P10635 1/20 0.40
CYP2C9 P11712 1/20 0.40
CYP2C19 P33261 1/20 0.40
L3MBTL1 Q9Y468 1/20 0.40
LMNA P02545 1/20 0.40
GRIN2D O15399 1/20 0.40
GRIN3B O60391 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6950820 0.93 ALDH1A1 (0.47) MEN1KMT2AALDH1A1KDM4EMAPK1
SCHEMBL6953001 0.92 MEN1 (0.56) MEN1KMT2ANPC1ALDH1A1KDM4E
SCHEMBL6958696 0.85 MEN1 (0.46) MEN1KMT2ANPC1KDM4EMAPK1
SCHEMBL6956012 0.85 TACR3 (0.43) MEN1KMT2ANPC1KDM4EMAPK1
SCHEMBL6959025 0.83 DRD2 (0.44) MEN1KMT2ANPC1KDM4EMAPK1
SCHEMBL6959021 0.83 CARM1 (0.45) MEN1KMT2ANPC1ALDH1A1KDM4E
SCHEMBL6958270 0.83 TACR1 (0.51) MEN1KMT2AALDH1A1KDM4EMAPK1
SCHEMBL6959388 0.81 TACR1 (0.51) MEN1KMT2AALDH1A1TACR3
SCHEMBL18782564 0.81 AKR1C3 (0.50) NPC1ALDH1A1HPGDSMN1; SMN2TACR3
SCHEMBL6954412 0.80 TACR3 (0.43) MEN1KMT2AKDM4EMAPK1HPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0993458-B1 3-BENZYLPIPERIDINE MERCK PATENT GMBH (DE) 2003-04-09 EP disclosed
US-6333339-B1 CENTRAL SYSTEM DISORDERS, SCHIZOPHRENIA AND COGNITION ACTIVATORS MERCK PATENT GELLSCHAFT MIT BESCHRANKTER (DE) 2001-12-25 US disclosed
EP-0993458-A1 3-BENZYLPIPERIDINE MERCK PATENT GmbH (DE) 2000-04-19 EP disclosed
WO-1998057953-A1 3-BENZYLPIPERIDINE MERCK PATENT GMBH (DE) 1998-12-23 WO disclosed