Imidazole

Imidazole

SCHEMBL6959692

C=CCCC(=O)C(c1ccccc1)(c1ccccc1)c1ccccc1.c1c[nH]cn1

nearest known ligand 0.36

Full drug profile on Sugi Atlas →

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.36
TSHR P16473 1/20 0.36
HTT P42858 1/20 0.35
FKBP5 Q13451 1/20 0.33
KDM4E B2RXH2 1/20 0.31
DAGLA Q9Y4D2 1/20 0.31
NPSR1 Q6W5P4 1/20 0.31
KMT2A Q03164 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8939183 0.83 ALDH1A1 (0.49) ALDH1A1TSHRHTTKDM4ENPSR1
Imidazole SCHEMBL4551598 0.74 ALDH1A1 (0.41) ALDH1A1FKBP5
Imidazole SCHEMBL28750264 0.72 MAPT (0.50) ALDH1A1FKBP5KDM4EKMT2A
Imidazole SCHEMBL2541492 0.71 ALDH1A1 (0.48) ALDH1A1FKBP5
Imidazole SCHEMBL29140670 0.71 MAPT (0.49) ALDH1A1FKBP5KDM4EKMT2A
Benzylic Acid SCHEMBL10563379 0.70 CYP2C9 (0.49) ALDH1A1HTTFKBP5NPSR1KMT2A
Imidazole SCHEMBL28904975 0.69 ALDH1A1 (0.54) ALDH1A1TSHRFKBP5KMT2A
Allylbenzene SCHEMBL27805393 0.68 ALDH1A1 (0.45) ALDH1A1TSHRFKBP5
Acrylic Acid SCHEMBL2459820 0.67 ALDH1A1 (0.56) ALDH1A1FKBP5
Acrylic Acid SCHEMBL9807323 0.67 ALDH1A1 (0.56) ALDH1A1FKBP5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1318996-A2 SUBSTITUTED IMIDAZOLES AS DUAL HISTAMINE H1 AND H3 AGONISTS OR ANTAGONISTS Schering Corporation (US) 2003-06-18 EP disclosed
EP-1318994-A2 SUBSTITUTED IMIDAZOLES AS DUAL HISTAMINE H1 AND H3 AGONISTS OR ANTAGONISTS Schering Corporation (US) 2003-06-18 EP disclosed
WO-2002044141-A2 SUBSTITUTED IMIDAZOLES AS DUAL HISTAMINE H1 AND H3 AGONISTS OR ANTAGONISTS SCHERING CORPORATION (US) 2002-06-06 WO disclosed
WO-2002024659-A2 SUBSTITUTED IMIDAZOLES AS DUAL HISTAMINE H1 AND H3 AGONISTS OR ANTGONISTS SCHERING CORPORATION (US) 2002-03-28 WO disclosed