SCHEMBL6960025

SCHEMBL6960025

CC(C)c1cc(Cc2nc3cccc(C#Cc4ccccn4)c3o2)cc(C(C)C)c1O

nearest known ligand 0.34

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GRM5 P41594 5/20 0.34
KCNH2 Q12809 2/20 0.34
DHFR P00374 1/20 0.34
ERN1 O75460 1/20 0.34
THRA P10827 1/20 0.34
THRB P10828 1/20 0.34
NPC1 O15118 3/20 0.33
RAB9A P51151 3/20 0.33
MEN1 O00255 2/20 0.33
KMT2A Q03164 2/20 0.33
PTGES O14684 1/20 0.31
AKR1C3 P42330 1/20 0.31
PTGDR2 Q9Y5Y4 1/20 0.31
HCRTR1 O43613 1/20 0.31
POLB P06746 1/20 0.31
ELANE P08246 1/20 0.31
LMNA P02545 1/20 0.30
TP53 P04637 1/20 0.30
SMN1; SMN2 Q16637 1/20 0.30
ACACB O00763 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6960215 0.85 GAA (0.36) GRM5KCNH2DHFRERN1MEN1
SCHEMBL6960207 0.76 DHFR (0.38) DHFRMEN1KMT2AELANELMNA
SCHEMBL6964996 0.74 PTGDR2 (0.38) GRM5KCNH2DHFRERN1NPC1
SCHEMBL103255 0.70 GRM5 (0.38) GRM5KCNH2ELANE
SCHEMBL102341 0.65 GRM5 (0.39) GRM5KCNH2TP53SMN1; SMN2
SCHEMBL7734764 0.64 DHFR (0.40) DHFRMEN1KMT2ALMNATP53
SCHEMBL102632 0.64 GRM5 (0.40) GRM5KCNH2ERN1NPC1RAB9A
SCHEMBL103358 0.62 GRM5 (0.42) GRM5KCNH2NPC1RAB9AELANE
SCHEMBL16004606 0.60 GRM5 (0.57) GRM5KCNH2
SCHEMBL30526535 0.60 GRM5 (0.57) GRM5KCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0785927-B1 NOVEL BENZOXAZOLES EURO CELTIQUE SA (LU) 2003-08-27 EP claimed