SCHEMBL6960347

SCHEMBL6960347

CN1CCCC1c1cncc(C#CC(C)(C)OC(=O)/C=C/C(=O)OC(C)(C)C#Cc2cncc(C3CCCN3C)c2)c1

nearest known ligand 0.55

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CHRNA3 P32297 8/20 0.55
CHRNB2 P17787 7/20 0.55
CHRNB4 P30926 6/20 0.55
CHRNA1 P02708 4/20 0.55
CHRNA4 P43681 4/20 0.55
CHRNA2 Q15822 4/20 0.55
CHRNB1 P11230 3/20 0.55
CHRNG P07510 2/20 0.55
CHRND Q07001 2/20 0.55
KDM4E B2RXH2 1/20 0.40
BLM P54132 1/20 0.40
ALOX15 P16050 1/20 0.40
CHRNB3 Q05901 2/20 0.39
ALDH1A1 P00352 2/20 0.39
CHRNA7 P36544 2/20 0.39
LMNA P02545 1/20 0.39
TDP1 Q9NUW8 1/20 0.39
HTR3E A5X5Y0 1/20 0.39
PSIP1 O75475 1/20 0.39
TRPA1 O75762 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6959278 0.82 CHRNA3 (0.64) CHRNA3CHRNB2CHRNB4CHRNA1CHRNA4
SCHEMBL6961453 0.81 CHRNA3 (0.55) CHRNA3CHRNB2CHRNB4CHRNA1CHRNA4
SCHEMBL6966231 0.80 CHRNA3 (0.54) CHRNA3CHRNB2CHRNB4CHRNA1CHRNA4
SCHEMBL6973016 0.80 CHRNA3 (0.53) CHRNA3CHRNB2CHRNB4CHRNA1CHRNA4
Fumaric Acid SCHEMBL6961573 0.78 CHRNB4 (0.59) CHRNA3CHRNB2CHRNB4CHRNA1CHRNA4
SCHEMBL6813669 0.78 CHRNA3 (0.64) CHRNA3CHRNB2CHRNB4CHRNA1CHRNA4
Fumaric Acid SCHEMBL6960624 0.77 CHRNB4 (0.57) CHRNA3CHRNB2CHRNB4CHRNA1CHRNA4
Fumaric Acid SCHEMBL6960621 0.77 CHRNB4 (0.57) CHRNA3CHRNB2CHRNB4CHRNA1CHRNA4
SCHEMBL6972915 0.76 CHRNB4 (0.72) CHRNA3CHRNB2CHRNB4CHRNA1CHRNA4
Altinicline SCHEMBL15253516 0.75 CHRNA3 (0.79) CHRNA3CHRNB2CHRNB4CHRNA1CHRNA4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0739342-B1 PYRIDINE MODULATORS OF ACETYLCHOLINE RECEPTORS MERCK & CO INC (US) 2003-08-27 EP disclosed