SCHEMBL6960446

SCHEMBL6960446

COc1cccc(N2CCN(C(=S)Nc3cc4ccccc4nc3OC)CC2)c1

nearest known ligand 0.63

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 2/20 0.60
MEN1 O00255 5/20 0.58
KMT2A Q03164 5/20 0.58
CYP3A4 P08684 2/20 0.58
CYP2C9 P11712 2/20 0.58
CYP2C19 P33261 2/20 0.58
CYP1A2 P05177 1/20 0.58
PHGDH O43175 4/20 0.58
PKM P14618 1/20 0.58
POLB P06746 3/20 0.57
LMNA P02545 3/20 0.56
MAPT P10636 4/20 0.53
GAA P10253 2/20 0.53
ALDH1A1 P00352 3/20 0.50
RAB9A P51151 1/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6652797 0.92 PHGDH (0.55) NPC1MEN1KMT2ACYP3A4CYP2C9
SCHEMBL6650903 0.90 KDM4E (0.59) NPC1MEN1KMT2ACYP3A4CYP2C9
SCHEMBL27467994 0.88 KMT2A (0.64) KMT2APOLBLMNAMAPTGAA
SCHEMBL6651512 0.87 PHGDH (0.52) MEN1KMT2ACYP3A4CYP2C19PHGDH
SCHEMBL6780801 0.86 MAPT (0.47) NPC1MEN1KMT2ACYP3A4CYP2C9
SCHEMBL6960635 0.86 PHGDH (0.54) MEN1KMT2ACYP3A4CYP2C9CYP2C19
SCHEMBL27556985 0.84 MEN1 (0.63) NPC1MEN1KMT2ACYP3A4CYP2C9
SCHEMBL6650534 0.82 PHGDH (0.59) NPC1MEN1KMT2ACYP3A4CYP2C9
SCHEMBL6965032 0.81 PHGDH (0.58) NPC1MEN1KMT2ACYP3A4CYP2C9
SCHEMBL6966994 0.81 KMT2A (0.55) KMT2APOLBLMNAMAPTGAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-100354271-C Piperazine derivatives and process for the preparation thereof SAMJIN PHARM CO LTD (KR) 2007-12-12 CN disclosed
EP-0850222-B1 PIPERAZINE DERIVATIVES AND PROCESS FOR THE PREPARATION THEREOF SAMJIN PHARM CO LTD (KR) 2003-05-28 EP disclosed
CN-1296477-A Piperazine derivatives and process for the preparation thereof SAMJIN PHARM CO LTD (KR) 2001-05-23 CN disclosed
US-6028195-A AN ANTITUMOR AGENT WITH VERY LOW TOXICITIES SAMJIN PHARMACEUTICAL CO., LTD. (KR) 2000-02-22 US disclosed
EP-0850222-A1 PIPERAZINE DERIVATIVES AND PROCESS FOR THE PREPARATION THEREOF Samjin Pharmaceutical Co., Ltd. (KR) 1998-07-01 EP disclosed
WO-1998000402-A1 PIPERAZINE DERIVATIVES AND PROCESS FOR THE PREPARATION THEREOF SAMJIN PHARMACEUTICAL CO., LTD. (KR) 1998-01-08 WO disclosed