SCHEMBL6965032

SCHEMBL6965032

COc1cc(OC)cc(N2CCN(C(=S)Nc3cc4ccccc4nc3C)CC2)c1

nearest known ligand 0.58

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
PHGDH O43175 5/20 0.58
MEN1 O00255 3/20 0.53
KMT2A Q03164 3/20 0.53
POLB P06746 2/20 0.53
CYP3A4 P08684 3/20 0.51
CYP2C19 P33261 2/20 0.51
HTT P42858 1/20 0.50
NPC1 O15118 2/20 0.49
GAA P10253 2/20 0.49
MAPT P10636 2/20 0.49
SMN1; SMN2 Q16637 1/20 0.49
PKM P14618 1/20 0.49
CYP2C9 P11712 2/20 0.48
ALDH1A1 P00352 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6652797 0.89 PHGDH (0.55) PHGDHMEN1KMT2APOLBCYP3A4
SCHEMBL6966237 0.88 PHGDH (0.56) PHGDHMEN1KMT2APOLBCYP3A4
SCHEMBL6956583 0.87 KMT2A (0.53) PHGDHKMT2APOLBGAAMAPT
SCHEMBL6960143 0.86 KMT2A (0.48) PHGDHMEN1KMT2APOLBGAA
SCHEMBL6651512 0.82 PHGDH (0.52) PHGDHMEN1KMT2APOLBCYP3A4
SCHEMBL6960446 0.81 NPC1 (0.60) PHGDHMEN1KMT2APOLBCYP3A4
SCHEMBL6960635 0.79 PHGDH (0.54) PHGDHMEN1KMT2APOLBCYP3A4
SCHEMBL6780801 0.79 MAPT (0.47) PHGDHMEN1KMT2APOLBCYP3A4
SCHEMBL6654161 0.78 PHGDH (0.60) PHGDHMEN1KMT2APOLBCYP3A4
SCHEMBL6562602 0.78 PHGDH (0.57) PHGDHMEN1KMT2APOLBCYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0850222-B1 PIPERAZINE DERIVATIVES AND PROCESS FOR THE PREPARATION THEREOF SAMJIN PHARM CO LTD (KR) 2003-05-28 EP disclosed
US-6028195-A AN ANTITUMOR AGENT WITH VERY LOW TOXICITIES SAMJIN PHARMACEUTICAL CO., LTD. (KR) 2000-02-22 US disclosed
EP-0850222-A1 PIPERAZINE DERIVATIVES AND PROCESS FOR THE PREPARATION THEREOF Samjin Pharmaceutical Co., Ltd. (KR) 1998-07-01 EP disclosed
WO-1998000402-A1 PIPERAZINE DERIVATIVES AND PROCESS FOR THE PREPARATION THEREOF SAMJIN PHARMACEUTICAL CO., LTD. (KR) 1998-01-08 WO disclosed