SCHEMBL6961827

SCHEMBL6961827

Nc1ccc(CCCC(=O)Nc2ccccc2)cc1

nearest known ligand 0.68

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM1A O60341 2/20 0.68
TRPV1 Q8NER1 1/20 0.66
HDAC1 Q13547 9/20 0.65
HDAC4 P56524 8/20 0.65
HDAC7 Q8WUI4 8/20 0.65
HDAC11 Q96DB2 8/20 0.65
HDAC8 Q9BY41 8/20 0.65
HDAC6 Q9UBN7 8/20 0.65
HDAC9 Q9UKV0 8/20 0.65
HDAC5 Q9UQL6 8/20 0.65
HDAC3 O15379 7/20 0.65
HDAC2 Q92769 7/20 0.65
HDAC10 Q969S8 7/20 0.65
MAPT P10636 2/20 0.63
HTT P42858 1/20 0.63
NPC1 O15118 2/20 0.59
RAB9A P51151 2/20 0.59
ALDH1A1 P00352 1/20 0.59
ALOX15 P16050 1/20 0.59
NFKB1 P19838 1/20 0.59

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL8392010 0.98 KDM1A (0.66) KDM1ATRPV1HDAC1HDAC4HDAC7
SCHEMBL8012743 0.89 TRPV1 (0.81) KDM1ATRPV1HDAC1HDAC4HDAC7
SCHEMBL17064271 0.86 KDM1A (0.58) KDM1ATRPV1HDAC1HDAC4HDAC7
SCHEMBL1064492 0.85 HDAC1 (0.74) HDAC1HDAC4HDAC7HDAC11HDAC8
SCHEMBL8244867 0.85 HDAC1 (0.74) HDAC1HDAC4HDAC7HDAC11HDAC8
SCHEMBL20508341 0.84 HDAC1 (0.69) KDM1ATRPV1HDAC1HDAC4HDAC7
SCHEMBL10198474 0.84 MAPT (0.77) TRPV1HDAC1HDAC4HDAC7HDAC11
SCHEMBL7636110 0.83 TRPV1 (0.77) KDM1ATRPV1HDAC1HDAC4HDAC7
SCHEMBL19501635 0.83 TRPV1 (0.77) KDM1ATRPV1HDAC1HDAC4HDAC7
SCHEMBL28099312 0.82 MAPT (0.74) KDM1ATRPV1HDAC1HDAC4HDAC7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0713483-B1 AMIDINE DERIVATIVES WITH NITRIC OXIDE SYNTHETASE ACTIVITIES ASTRAZENECA AB (SE) 2003-01-15 EP disclosed
US-6030985-A Amidine derivatives with nitric oxide synthetase activities ASTRA AKTIEBOLAG (SE) 2000-02-29 US disclosed
US-5807885-A Amidine derivatives with nitric oxide synthetase activities ASTRA AKTIEBOLAG (SE) 1998-09-15 US disclosed
EP-0713483-A1 AMIDINE DERIVATIVES WITH NITRIC OXIDE SYNTHETASE ACTIVITIES Astra Aktiebolag (SE) 1996-05-29 EP disclosed
WO-1995005363-A1 AMIDINE DERIVATIVES WITH NITRIC OXIDE SYNTHETASE ACTIVITIES ASTRA AKTIEBOLAG (SE) 1995-02-23 WO disclosed