SCHEMBL6962115

SCHEMBL6962115

CC(C)c1nc(C(O)Cc2ccccc2)[nH]c1Sc1cc(F)cc(F)c1

nearest known ligand 0.32

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
ADRB2 P07550 4/20 0.32
PYGL P06737 2/20 0.32
MAPK14 Q16539 1/20 0.31
LMNA P02545 1/20 0.31
TRPA1 O75762 1/20 0.31
IDO1 P14902 2/20 0.31
CAPN1 P07384 1/20 0.30
DHFR P00374 1/20 0.30
POLB P06746 1/20 0.30
HPGD P15428 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6961240 0.90 MAPK14 (0.34) MAPK14CAPN1POLB
SCHEMBL6960986 0.90 GSK3B (0.32)
SCHEMBL6965426 0.89 GPR84 (0.33) MAPK14CAPN1
SCHEMBL7087539 0.89 ADRB2 (0.34) ADRB2
SCHEMBL6969546 0.88 IDO1 (0.36) MAPK14IDO1
SCHEMBL6970755 0.88 ADRB2 (0.38) ADRB2
SCHEMBL6967546 0.87 IDO1 (0.38) ADRB2LMNATRPA1IDO1CAPN1
SCHEMBL6966853 0.86 TDP1 (0.33) ADRB2PYGLTRPA1IDO1CAPN1
SCHEMBL6969061 0.86
SCHEMBL6973516 0.86 PTPRA (0.33) MAPK14

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0786455-B1 IMIDAZOLE DERIVATIVE SHIONOGI & CO (JP) 2003-12-03 EP disclosed
US-6147097-A METHOD FOR TREATING AIDS SHIONOGI & CO., LTD. (JP) 2000-11-14 US disclosed
US-5910506-A IMIDAZOLE DERIVATIVES, E.G.5-(3,5-DICHLOROPHENYLTHIO)-1,2-DIMETHYL-4-ISOPROPYL-1H-IMIDAZOLE; VIRICIDES; AIDS; NONTOXIC SHIONOGI & CO., LTD. (JP) 1999-06-08 US disclosed
EP-0786455-A1 IMIDAZOLE DERIVATIVE SHIONOGI & CO., LTD. (JP) 1997-07-30 EP disclosed