SCHEMBL6963015

SCHEMBL6963015

CCC/C=C(/C([O])=O)c1ccccc1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 5/20 0.48
CYP1A2 P05177 4/20 0.48
TSHR P16473 4/20 0.48
ALDH1A1 P00352 3/20 0.48
CES2 O00748 5/20 0.43
CES1 P23141 5/20 0.43
CYP2C9 P11712 4/20 0.42
CYP2C19 P33261 4/20 0.42
MAPK1 P28482 1/20 0.42
SMN1; SMN2 Q16637 1/20 0.42
LMNA P02545 3/20 0.42
AKR1C1 Q04828 1/20 0.40
CYP2D6 P10635 2/20 0.39
MTNR1A P48039 1/20 0.39
MTNR1B P49286 1/20 0.39
MAPT P10636 3/20 0.38
HTT P42858 2/20 0.38
NPSR1 Q6W5P4 2/20 0.38
L3MBTL1 Q9Y468 1/20 0.38
KDM4E B2RXH2 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6973235 0.89 CYP1A2 (0.47) CYP3A4CYP1A2TSHRALDH1A1CES2
SCHEMBL8041709 0.87 AKR1C1 (0.50) CYP3A4CYP1A2TSHRALDH1A1CES2
SCHEMBL8041704 0.87 AKR1C1 (0.50) CYP3A4CYP1A2TSHRALDH1A1CES2
SCHEMBL6259485 0.87 AKR1C1 (0.50) CYP3A4CYP1A2TSHRALDH1A1CES2
SCHEMBL14763931 0.85 CES2 (0.45) CYP3A4CYP1A2TSHRALDH1A1CES2
SCHEMBL6971325 0.85 CES1 (0.44) CYP3A4TSHRALDH1A1CES2CES1
SCHEMBL6209765 0.84 CYP3A4 (0.43) CYP3A4CYP1A2TSHRALDH1A1CES2
SCHEMBL2109360 0.77 SMN1; SMN2 (0.53) CYP3A4CYP1A2ALDH1A1SMN1; SMN2MAPT
SCHEMBL8157814 0.76 CES2 (0.47) CYP3A4CYP1A2TSHRALDH1A1CES2
SCHEMBL524133 0.76 CES2 (0.47) CYP3A4CYP1A2TSHRALDH1A1CES2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1329160-A2 4-ACYLAMINOPYRAZOLE DERIVATIVES Sankyo Company, Limited (JP) 2003-07-23 EP disclosed