SCHEMBL6964051

SCHEMBL6964051

CCn1c(CCOC(C)=O)nc(C(C)C)c1Sc1cccc([N+](=O)[O-])c1

nearest known ligand 0.35

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
IRAK4 Q9NWZ3 1/20 0.35
CYP2C9 P11712 5/20 0.35
CYP2C19 P33261 5/20 0.35
CYP1A2 P05177 4/20 0.35
CYP3A4 P08684 4/20 0.35
MAPT P10636 2/20 0.35
CACNA1F O60840 3/20 0.35
CACNA1D Q01668 3/20 0.35
CACNA1S Q13698 3/20 0.35
CACNA1C Q13936 3/20 0.35
CYP2D6 P10635 2/20 0.35
RECQL P46063 1/20 0.35
KMT2A Q03164 4/20 0.34
MEN1 O00255 3/20 0.34
LMNA P02545 2/20 0.34
TSHR P16473 1/20 0.34
NFKB1 P19838 1/20 0.34
THPO P40225 1/20 0.34
HSP90AA1 P07900 1/20 0.34
CFTR P13569 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6971930 0.93 CYP2C9 (0.36) IRAK4CYP2C9CYP2C19CYP1A2CYP3A4
SCHEMBL6973804 0.92 CACNA1F (0.36) IRAK4CYP2C9CYP2C19CYP1A2CYP3A4
SCHEMBL7083140 0.92 CYP2C9 (0.39) IRAK4CYP2C9CYP2C19CYP1A2CYP3A4
SCHEMBL6971525 0.89 NPC1 (0.36) CYP2C9CYP2C19CYP1A2CYP3A4MAPT
SCHEMBL7086066 0.88 KMT2A (0.36) CYP2C9CYP2C19MAPTCYP2D6RECQL
SCHEMBL6964484 0.87 CACNA1F (0.36) IRAK4CYP2C9CYP2C19CYP1A2CYP3A4
SCHEMBL7080984 0.87 LMNA (0.38) IRAK4CYP2C9CYP2C19CYP1A2CYP3A4
SCHEMBL6972280 0.87 CFTR (0.40) CYP1A2CYP3A4MAPTKMT2AMEN1
SCHEMBL6971341 0.86 CYP2C9 (0.38) IRAK4CYP2C9CYP2C19CYP1A2CYP3A4
SCHEMBL6971348 0.86 CYP2C9 (0.38) IRAK4CYP2C9CYP2C19CYP1A2CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0786455-B1 IMIDAZOLE DERIVATIVE SHIONOGI & CO (JP) 2003-12-03 EP disclosed
US-6147097-A METHOD FOR TREATING AIDS SHIONOGI & CO., LTD. (JP) 2000-11-14 US disclosed
US-5910506-A IMIDAZOLE DERIVATIVES, E.G.5-(3,5-DICHLOROPHENYLTHIO)-1,2-DIMETHYL-4-ISOPROPYL-1H-IMIDAZOLE; VIRICIDES; AIDS; NONTOXIC SHIONOGI & CO., LTD. (JP) 1999-06-08 US disclosed