Bicarbonate

Bicarbonate

SCHEMBL6964764

Brc1ccsc1Br.O=C(O)O

nearest known ligand 0.40

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Known targets — ChEMBL curated mechanism

GSK3AGSK3BIMPA1

The experimentally established mechanism targets of Bicarbonate. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
POLB P06746 2/20 0.40
TSHR P16473 1/20 0.37
DAO P14920 3/20 0.34
GPR35 Q9HC97 3/20 0.33
SLC6A4 P31645 1/20 0.33
SLC6A3 Q01959 1/20 0.33
PTPRC P08575 1/20 0.33
PTPRG P23470 1/20 0.33
MAPT P10636 2/20 0.33
NPC1 O15118 1/20 0.33
PKM P14618 1/20 0.33
RAB9A P51151 1/20 0.33
NPSR1 Q6W5P4 1/20 0.33
RXFP1 Q9HBX9 1/20 0.33
ALDH1A1 P00352 4/20 0.32
MEN1 O00255 2/20 0.32
KMT2A Q03164 2/20 0.32
HDAC1 Q13547 1/20 0.32
MAPK1 P28482 1/20 0.32
KDM4E B2RXH2 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL134132 0.87
Formic Acid SCHEMBL27906489 0.83 POLB (0.39) POLB
SCHEMBL399760 0.73
SCHEMBL7045346 0.70 POLB (0.49) POLBPTPRCPTPRGNPSR1ALDH1A1
SCHEMBL1992958 0.69 PTPN2 (0.43) TSHRMAPTNPC1PKMRAB9A
SCHEMBL2684375 0.69 SLC6A4 (0.44) SLC6A4SLC6A3MAPTALDH1A1MEN1
SCHEMBL3418797 0.69 POLB (0.40) POLBDAOGPR35PTPRCPTPRG
SCHEMBL1009157 0.69 PTPN2 (0.43) POLBMAPTNPC1RAB9AMEN1
SCHEMBL507698 0.67
SCHEMBL621972 0.67

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0676395-B1 Substituted N-heteroaroylguanidines, as inhibitors of sodium-hydrogen exchange, as antiarrhythmic agents and as inhibitors of the proliferation of cells HOECHST AG (DE) 2003-09-03 EP disclosed
EP-0755185-A1 MICROBICIDAL AGENTS BASED ON DIBROMO-THIOPHENE-CARBOXYLIC ACID DERIVATIVES BAYER AG (DE) 1997-01-29 EP disclosed
WO-1995027397-A1 MICROBICIDAL AGENTS BASED ON DIBROMO-THIOPHENE-CARBOXYLIC ACID DERIVATIVES BAYER AKTIENGESELLSCHAFT (DE) 1995-10-19 WO disclosed
EP-0676395-A2 Substituted N-heteroaroylguanidines, as inhibitors of sodium-hydrogen exchange, as antiarrhythmic agents and as inhibitors of the proliferation of cells HOECHST AKTIENGESELLSCHAFT (DE) 1995-10-11 EP disclosed