SCHEMBL6965067

SCHEMBL6965067

O=C1NC(=O)C(Cc2cnc3cc(OCc4ccccc4)ccc3c2)O1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 2/20 0.46
IP6K1 Q92551 1/20 0.42
MAOB P27338 9/20 0.42
MAOA P21397 5/20 0.42
NPC1 O15118 2/20 0.42
MEN1 O00255 1/20 0.42
CA12 O43570 1/20 0.42
CA1 P00915 1/20 0.42
CA2 P00918 1/20 0.42
CA3 P07451 1/20 0.42
CA4 P22748 1/20 0.42
CA6 P23280 1/20 0.42
CA7 P43166 1/20 0.42
MTNR1A P48039 1/20 0.42
KMT2A Q03164 1/20 0.42
CA9 Q16790 1/20 0.42
CA14 Q9ULX7 1/20 0.42
ALOX5 P09917 1/20 0.41
PDGFRB P09619 1/20 0.41
PDGFRA P16234 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7987732 0.81 MEN1 (0.49) MAOBMAOAMEN1KMT2A
SCHEMBL29602962 0.79 FFAR1 (0.59) CYP3A4
SCHEMBL377641 0.79 FFAR1 (0.59) CYP3A4
SCHEMBL6959497 0.78 MAOB (0.55) CYP3A4MAOBMAOAALOX5
SCHEMBL377642 0.77 CYP3A4 (0.46) CYP3A4IP6K1MAOBMAOANPC1
SCHEMBL8172462 0.77 MAOB (0.48) CYP3A4IP6K1MAOBMAOANPC1
SCHEMBL8315754 0.75 FFAR1 (0.48) MAOBMAOAMEN1KMT2A
SCHEMBL6956120 0.74 FFAR1 (0.63)
SCHEMBL18571362 0.73 CYP3A4 (0.61) CYP3A4MAOBNPC1ALOX5PDGFRB
SCHEMBL6958784 0.72 FFAR1 (0.58) CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0787725-B1 QUINOLINE DERIVATIVE NIPPON CHEMIPHAR CO (JP) 2003-04-23 EP disclosed
US-5693651-A HYPOGLYCEMIC AGENTS NIPPON CHEMIPHAR CO., LTD. (JP) 1997-12-02 US disclosed
EP-0787725-A1 QUINOLINE DERIVATIVE NIPPON CHEMIPHAR CO., LTD. (JP) 1997-08-06 EP disclosed