SCHEMBL7987732

SCHEMBL7987732

O=C1NC(=O)C(Cc2ccc(OCc3ccccc3)cc2)O1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 1/20 0.49
KMT2A Q03164 1/20 0.49
KDM4C Q9H3R0 1/20 0.49
FFAR1 O14842 3/20 0.47
LMNA P02545 2/20 0.45
GRM2 Q14416 1/20 0.45
MMP2 P08253 1/20 0.45
MMP13 P45452 1/20 0.45
MAOB P27338 3/20 0.45
MAOA P21397 2/20 0.45
GSTP1 P09211 1/20 0.44
PPARA Q07869 1/20 0.44
BCHE P06276 1/20 0.44
PPARG P37231 1/20 0.44
CYP1A2 P05177 1/20 0.44
PTGS1 P23219 1/20 0.44
SLC6A2 P23975 1/20 0.44
CYP2C19 P33261 1/20 0.44
PTGS2 P35354 1/20 0.44
SLC6A3 Q01959 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8315754 0.94 FFAR1 (0.48) MEN1KMT2AKDM4CFFAR1LMNA
SCHEMBL12521895 0.89 CTSK (0.46) KMT2AFFAR1MAOBMAOAPPARG
SCHEMBL8889741 0.87 FFAR1 (0.48) FFAR1GRM2MMP2MMP13MAOB
SCHEMBL8181635 0.85 CA2 (0.41) MEN1KMT2AFFAR1MMP2MMP13
SCHEMBL8888011 0.84 LTA4H (0.49) FFAR1GRM2BCHEFFAR4HPGD
SCHEMBL8172462 0.83 MAOB (0.48) MEN1KMT2ALMNAMAOBMAOA
SCHEMBL8888854 0.83 MGLL (0.50) FFAR1GRM2BCHEFFAR4HPGD
SCHEMBL8890354 0.83 MGLL (0.50) FFAR1GRM2BCHEFFAR4HPGD
SCHEMBL8888505 0.83 MGLL (0.50) FFAR1GRM2BCHEFFAR4HPGD
SCHEMBL8312946 0.81 CYP4F2 (0.39) MEN1KMT2AFFAR1PPARAPPARG

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6288096-B1 ANTIDIABETIC AGENTS, HYPOTENSIVE AGENTS, AND ANTICHOLESTEROL AGENTS ASTRAZENECA AB (SE) 2001-09-11 US disclosed
EP-0991632-A1 NEW THIAZOLIDINEDIONE, OXAZOLIDINEDIONE AND OXADIAZOLIDINEDIONE DERIVATIVES Astra Aktiebolag (SE) 2000-04-12 EP disclosed
WO-1998057941-A1 NEW THIAZOLIDINEDIONE, OXAZOLIDINEDIONE AND OXADIAZOLIDINEDIONE DERIVATIVES ASTRA AKTIEBOLAG (SE) 1998-12-23 WO disclosed
US-5391565-A Hypoglycemic agents; antilipemic agents; hypotensive agents BEECHAN GROUP P.L.C. (GB) 1995-02-21 US disclosed