SCHEMBL6965295

SCHEMBL6965295

CCCCN1CCN(C(Cc2ccc(C#N)cc2)c2cnc[nH]2)C(c2ccccc2C)C1=O

nearest known ligand 0.36

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
CYP19A1 P11511 2/20 0.36
FNTA P49354 14/20 0.35
FNTB P49356 14/20 0.35
KCNH2 Q12809 2/20 0.34
PGGT1B P53609 5/20 0.33
CYP11B1 P15538 1/20 0.32
CYP11B2 P19099 1/20 0.32
MC4R P32245 2/20 0.31
MC1R Q01726 2/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5758460 0.94 FNTA (0.38) CYP19A1FNTAFNTBKCNH2PGGT1B
SCHEMBL4405093 0.80 FNTA (0.40) CYP19A1FNTAFNTBKCNH2PGGT1B
SCHEMBL2381616 0.77 FNTA (0.47) CYP19A1FNTAFNTBKCNH2PGGT1B
SCHEMBL445939 0.74 FNTA (0.51) CYP19A1FNTAFNTBPGGT1BMC4R
SCHEMBL5131468 0.74 FNTA (0.51) CYP19A1FNTAFNTBPGGT1BMC4R
Hydrochloric Acid SCHEMBL8541088 0.73 FNTA (0.51) CYP19A1FNTAFNTBPGGT1BMC4R
Hydrochloric Acid SCHEMBL8160943 0.73 FNTA (0.51) CYP19A1FNTAFNTBPGGT1BMC4R
SCHEMBL3517007 0.73 FNTA (0.50) CYP19A1FNTAFNTBKCNH2PGGT1B
Trifluoroacetic Acid SCHEMBL8162228 0.73 FNTA (0.43) CYP19A1FNTAFNTBKCNH2PGGT1B
SCHEMBL3687066 0.71 FNTA (0.59) CYP19A1FNTAFNTBKCNH2PGGT1B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1226119-A4 TYROSINE KINASE INHIBITORS MERCK & CO INC (US) 2003-04-09 EP disclosed
EP-1226119-A2 TYROSINE KINASE INHIBITORS MERCK & CO. INC. (US) 2002-07-31 EP disclosed
WO-2001028993-A2 TYROSINE KINASE INHIBITORS MERCK & CO. INC. (US) 2001-04-26 WO disclosed