SCHEMBL6965668

SCHEMBL6965668

Cc1ccc([N+](=O)[O-])c(C)c1C1OCCO1

nearest known ligand 0.45

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.45
TSHR P16473 7/20 0.43
SMN1; SMN2 Q16637 2/20 0.43
TDP1 Q9NUW8 1/20 0.43
HSD17B10 Q99714 1/20 0.38
KMT2A Q03164 2/20 0.38
HTT P42858 1/20 0.38
CYP3A4 P08684 2/20 0.38
RECQL P46063 1/20 0.38
GAA P10253 1/20 0.36
KDM4E B2RXH2 1/20 0.36
MAPT P10636 1/20 0.36
MEN1 O00255 1/20 0.36
HPGD P15428 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL25993283 0.77 NSD2 (0.33)
SCHEMBL20328777 0.71 TSHR (0.53) ALDH1A1TSHRHSD17B10KMT2AHTT
SCHEMBL16740703 0.71 ATM (0.40) ALDH1A1TSHRSMN1; SMN2TDP1KMT2A
SCHEMBL3192674 0.70 TSHR (0.65) ALDH1A1TSHRSMN1; SMN2TDP1HSD17B10
SCHEMBL6973683 0.70 NSD2 (0.40) ALDH1A1TSHRTDP1CYP3A4
SCHEMBL7407826 0.70 TUBB4A (0.44) ALDH1A1TDP1KMT2AHTTMAPT
SCHEMBL9719281 0.70 TDP1 (0.71) ALDH1A1TSHRSMN1; SMN2TDP1HSD17B10
SCHEMBL30503599 0.70 TDP1 (0.71) ALDH1A1TSHRSMN1; SMN2TDP1HSD17B10
SCHEMBL1265167 0.70 TDP1 (0.54) ALDH1A1TSHRSMN1; SMN2TDP1HSD17B10
SCHEMBL10702744 0.69 TXNRD1 (0.60) ALDH1A1SMN1; SMN2KMT2AHTTCYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-1145623-C Imidazole derivatives - 2004-04-14 CN disclosed
EP-0797575-B1 IMIDAZOLE DERIVATIVES AS PROTEIN KINASE INHIBITORS IN PARTICULAR EGF-R TYROSINE KINASE HOFFMANN LA ROCHE (CH) 2003-10-15 EP disclosed
US-5959113-A REACTING A DIKETONE DERIVATIVE WITH AN ALDEHYDE DERIVATIVE; ADMINISTERING TO TREAT ATHEROSCLEROSIS, PSORIASIS, ALOPECIA AND TUMORS HOFFMANN-LA ROCHE INC. (US) 1999-09-28 US disclosed
CN-1175252-A Imidazole derivatives as protein kinase inhibitors in particular egf-rthyrosine kinase HOFFMANN LA ROCHE (CH) 1998-03-04 CN disclosed
EP-0797575-A1 IMIDAZOLE DERIVATIVES AS PROTEIN KINASE INHIBITORS IN PARTICULAR EGF-R TYROSINE KINASE F. HOFFMANN-LA ROCHE AG (CH) 1997-10-01 EP disclosed
WO-1996018626-A1 IMIDAZOLE DERIVATIVES AS PROTEIN KINASE INHIBITORS IN PARTICULAR EGF-R TYROSINE KINASE F. HOFFMANN-LA ROCHE AG (CH) 1996-06-20 WO disclosed