SCHEMBL6965853

SCHEMBL6965853

COc1ccc(F)c(CCNC(=S)Nc2ncc[nH]2)c1F

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 8/20 0.41
MEN1 O00255 6/20 0.41
GAA P10253 5/20 0.39
MAPT P10636 5/20 0.38
ADRA2A P08913 1/20 0.37
ADRA2C P18825 1/20 0.37
ADRA1D P25100 1/20 0.37
ADRA1A P35348 1/20 0.37
ADRA1B P35368 1/20 0.37
ALOX12 P18054 5/20 0.37
CYP1A2 P05177 1/20 0.37
CYP3A4 P08684 1/20 0.37
CYP2D6 P10635 1/20 0.37
CYP2C19 P33261 1/20 0.37
LMNA P02545 2/20 0.37
NPSR1 Q6W5P4 1/20 0.37
ALDH1A1 P00352 2/20 0.36
POLB P06746 1/20 0.36
MC4R P32245 1/20 0.36
SMN1; SMN2 Q16637 2/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6950698 0.91 KMT2A (0.42) KMT2AMEN1GAAMAPTALOX12
SCHEMBL6962193 0.87 GAA (0.44) KMT2AMEN1GAAMAPTALOX12
SCHEMBL6962622 0.83 GAA (0.45) KMT2AMEN1GAAMAPTALOX12
SCHEMBL6954353 0.82 RAB9A (0.42) KMT2AMEN1MAPTALOX12CYP1A2
SCHEMBL6964342 0.81 MAPT (0.41) KMT2AMEN1GAAMAPTADRA2A
SCHEMBL6957231 0.80 KMT2A (0.47) KMT2AMEN1GAAMAPTCYP1A2
SCHEMBL6958688 0.80 NPC1 (0.48) KMT2AMEN1GAAMAPTLMNA
SCHEMBL6957993 0.80 POLB (0.57) KMT2AMEN1GAAMAPTALOX12
SCHEMBL6954180 0.79 PTGES (0.38) KMT2AMEN1GAAMAPTALOX12
SCHEMBL6955550 0.79 KDM4E (0.49) KMT2AMEN1GAAMAPTCYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0540143-B1 Compounds and methods for inhibition of HIV and related viruses MEDIVIR AB (SE) 2003-02-05 EP disclosed
US-5714503-A Compounds and methods for inhibition of HIV and related viruses MEDIVIR AB (SE) 1998-02-03 US disclosed
US-5658907-A THIOUREA VIRICIDES MEDIVIR A/B (SE) 1997-08-19 US disclosed
US-5593993-A VIRICIDES FOR HTLV TREATMENT OF AIDS MEDIVIR AB (SE) 1997-01-14 US disclosed
EP-0540143-A2 Compounds and methods for inhibition of HIV and related viruses Medivir Aktiebolag (SE) 1993-05-05 EP disclosed