SCHEMBL696596

SCHEMBL696596

CC(C)(CS(=O)(=O)c1ccc(Cl)cc1Cl)C(=O)[C@@H]1C[C@@H](C(=O)O)N(C2CC2(C#N)C(N)=O)C1

nearest known ligand 0.33

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
LGMN Q99538 1/20 0.33
CTSS P25774 11/20 0.33
CTSL P07711 7/20 0.33
NOTUM Q6P988 1/20 0.32
KDM4E B2RXH2 1/20 0.32
CTSK P43235 1/20 0.31
TRPV4 Q9HBA0 4/20 0.31
CTSB P07858 1/20 0.31
DPP4 P27487 1/20 0.30
FAP Q12884 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL695622 0.91 CTSS (0.37) CTSSCTSLCTSKCTSB
SCHEMBL694304 0.87 CTSS (0.42) CTSSCTSLCTSKCTSB
SCHEMBL693779 0.83 CTSL (0.36) CTSSCTSLCTSKCTSB
SCHEMBL695487 0.83 CTSS (0.44) CTSSCTSLCTSKCTSB
Hydrochloric Acid SCHEMBL695250 0.82 CTSS (0.43) CTSSCTSLCTSKCTSB
SCHEMBL696530 0.78 CTSS (0.39) CTSSCTSLCTSKCTSB
Hydrochloric Acid SCHEMBL695707 0.77 CTSS (0.39) CTSSCTSLCTSKCTSB
SCHEMBL697241 0.76 CTSL (0.37) CTSSCTSLCTSB
SCHEMBL695657 0.75 CTSS (0.38) CTSSCTSLCTSKCTSB
SCHEMBL695639 0.75 CTSS (0.39) CTSSCTSLCTSB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2421826-A1 PROLINE DERIVATIVES AS CATHEPSIN INHIBITORS F. Hoffmann-La Roche AG (CH) 2012-02-29 EP disclosed