SCHEMBL6966027

SCHEMBL6966027

CC(C)C(c1ccccn1)c1nc(COC(N)=O)[nH]c1Sc1cc(Cl)cc(Cl)c1

nearest known ligand 0.33

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
XIAP P98170 1/20 0.33
BIRC2 Q13490 1/20 0.33
CACNA1B Q00975 1/20 0.32
PARP1 P09874 2/20 0.31
PARP3 Q9Y6F1 1/20 0.31
NPC1 O15118 1/20 0.31
RAB9A P51151 1/20 0.31
MAPT P10636 1/20 0.30
NPSR1 Q6W5P4 1/20 0.30
RHEB Q15382 1/20 0.30
MEN1 O00255 1/20 0.30
GAA P10253 1/20 0.30
KMT2A Q03164 1/20 0.30
SMN1; SMN2 Q16637 1/20 0.30
CYP1A2 P05177 1/20 0.30
CYP3A4 P08684 1/20 0.30
CYP2C9 P11712 1/20 0.30
CYP2C19 P33261 1/20 0.30
L3MBTL1 Q9Y468 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6975006 0.85 CXCR4 (0.33) XIAPBIRC2MAPTNPSR1CYP2C9
SCHEMBL6967039 0.85 KCNA5 (0.32) XIAPBIRC2PARP1PARP3MAPT
SCHEMBL5853041 0.85 GSK3B (0.31)
SCHEMBL6960435 0.84 HCAR2 (0.31) RAB9ACYP2C9L3MBTL1
SCHEMBL6957035 0.83 KCNA5 (0.35) GAA
SCHEMBL6559014 0.82 TYMS (0.32) MAPTCYP1A2CYP3A4CYP2C9CYP2C19
SCHEMBL8109045 0.80 PDE2A (0.32)
SCHEMBL5852656 0.76 GSK3B (0.32)
SCHEMBL6973398 0.76
SCHEMBL6971688 0.75 GSK3B (0.31) MAPTGAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0786455-B1 IMIDAZOLE DERIVATIVE SHIONOGI & CO (JP) 2003-12-03 EP disclosed
US-6147097-A METHOD FOR TREATING AIDS SHIONOGI & CO., LTD. (JP) 2000-11-14 US disclosed
US-5910506-A IMIDAZOLE DERIVATIVES, E.G.5-(3,5-DICHLOROPHENYLTHIO)-1,2-DIMETHYL-4-ISOPROPYL-1H-IMIDAZOLE; VIRICIDES; AIDS; NONTOXIC SHIONOGI & CO., LTD. (JP) 1999-06-08 US disclosed
EP-0786455-A1 IMIDAZOLE DERIVATIVE SHIONOGI & CO., LTD. (JP) 1997-07-30 EP disclosed