SCHEMBL6966049

SCHEMBL6966049

C[CH]C(=O)OC(C)c1ccccc1

nearest known ligand 0.69

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HCAR2 Q8TDS4 1/20 0.69
ALDH1A1 P00352 2/20 0.42
TP53 P04637 1/20 0.42
HSD17B10 Q99714 1/20 0.42
KMT2A Q03164 1/20 0.41
FFAR1 O14842 1/20 0.41
LPAR1 Q92633 2/20 0.40
LPAR3 Q9UBY5 1/20 0.40
CYP3A4 P08684 1/20 0.40
LTB4R Q15722 2/20 0.39
LTB4R2 Q9NPC1 2/20 0.39
GABRA1 P14867 1/20 0.39
GABRG2 P18507 1/20 0.39
GABRB3 P28472 1/20 0.39
GABRA5 P31644 1/20 0.39
GABRA3 P34903 1/20 0.39
GABRA2 P47869 1/20 0.39
GABRA4 P48169 1/20 0.39
GABRA6 Q16445 1/20 0.39
CYP2D6 P10635 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL573375 0.86 HCAR2 (0.89) HCAR2ALDH1A1TP53HSD17B10KMT2A
SCHEMBL10339803 0.86 HCAR2 (0.89) HCAR2ALDH1A1TP53HSD17B10KMT2A
SCHEMBL1845408 0.85 HCAR2 (0.75) HCAR2ALDH1A1TP53HSD17B10KMT2A
SCHEMBL1845412 0.85 HCAR2 (0.75) HCAR2ALDH1A1TP53HSD17B10KMT2A
SCHEMBL10638822 0.85 HCAR2 (0.69) HCAR2ALDH1A1TP53HSD17B10KMT2A
SCHEMBL10632315 0.85 HCAR2 (0.69) HCAR2ALDH1A1TP53HSD17B10KMT2A
SCHEMBL10638828 0.85 HCAR2 (0.69) HCAR2ALDH1A1TP53HSD17B10KMT2A
SCHEMBL41557 0.83 HCAR2 (0.67) HCAR2ALDH1A1TP53HSD17B10KMT2A
SCHEMBL28863896 0.83 HCAR2 (0.67) HCAR2ALDH1A1TP53HSD17B10KMT2A
SCHEMBL8869433 0.82 ESR1 (0.49) HCAR2ALDH1A1KMT2ACYP3A4CYP2D6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 9 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1329160-A2 4-ACYLAMINOPYRAZOLE DERIVATIVES Sankyo Company, Limited (JP) 2003-07-23 EP disclosed
US-5691341-A ANTILEUKEMIA AGENT OTSUKA PHARMACEUTICAL CO., LTD. (JP) 1997-11-25 US disclosed
US-5670563-A ORGANOTIN COMPOUND, PHOSPHORUS COMPOUND CIBA-SPECIALTY CHEMICALS CORPORATION (US) 1997-09-23 US disclosed
US-5639770-A SUPEROXIDE INHIBITOR OTSUKA PHARMACEUTICAL CO., LTD. (JP) 1997-06-17 US disclosed
US-5464833-A Anticarcinogenic agents, antiretrovirus agents or autoimmune diseases OTSUKA PHARMACEUTICAL CO., LTD. (JP) 1995-11-07 US disclosed
EP-0623598-A1 APOPTOSIS REGULATOR OTSUKA PHARMACEUTICAL CO., LTD. (JP) 1994-11-09 EP disclosed
US-5358949-A Carbostyril derivatives and salts thereof and anti-arrhythmic agents containing the carbostyril derivatives OTSUKA PHARMACEUTICAL CO., LTD. (JP) 1994-10-25 US disclosed
EP-0600092-A1 THIAZOLE DERIVATIVE OTSUKA PHARMACEUTICAL CO., LTD. (JP) 1994-06-08 EP disclosed
EP-0236140-A2 Carbostyril derivatives and salts thereof and anti-arrhythmic agents containing the carbostyril derivatives OTSUKA PHARMACEUTICAL CO., LTD. (JP) 1987-09-09 EP disclosed