SCHEMBL6966936

SCHEMBL6966936

O=S(=O)(c1ccc2nc3c(nc2c1)-c1cccc2cccc-3c12)c1cccc2cnccc12

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 2/20 0.45
HTR6 P50406 1/20 0.42
PRKD3 O94806 7/20 0.40
PRKCG P05129 7/20 0.40
PRKCB P05771 7/20 0.40
PRKCA P17252 7/20 0.40
PRKCH P24723 7/20 0.40
PRKCI P41743 7/20 0.40
PRKCE Q02156 7/20 0.40
PRKCQ Q04759 7/20 0.40
PRKCZ Q05513 7/20 0.40
PRKCD Q05655 7/20 0.40
PRKD1 Q15139 7/20 0.40
CYP3A4 P08684 6/20 0.40
PRKACA P17612 5/20 0.40
PRKACG P22612 5/20 0.40
PRKACB P22694 5/20 0.40
CYP2D6 P10635 5/20 0.40
MEN1 O00255 4/20 0.40
KMT2A Q03164 4/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6959990 0.85 TDP1 (0.52) CYP1A2HTR6PRKD3PRKCGPRKCB
SCHEMBL6968263 0.83 HTR6 (0.47) CYP1A2HTR6PRKD3PRKCGPRKCB
SCHEMBL6962780 0.83 PRKD3 (0.41) CYP1A2PRKD3PRKCGPRKCBPRKCA
SCHEMBL6966707 0.81 HTR6 (0.43) CYP1A2HTR6PRKD3PRKCGPRKCB
SCHEMBL6966099 0.81 HTR6 (0.48) CYP1A2HTR6PRKD3PRKCGPRKCB
SCHEMBL6958305 0.81 HTR6 (0.45) CYP1A2HTR6PRKD3PRKCGPRKCB
SCHEMBL6967123 0.74 CYP3A4 (0.50) CYP1A2HTR6PRKD3PRKCGPRKCB
SCHEMBL6967362 0.74 CYP3A4 (0.59) CYP1A2PRKD3PRKCGPRKCBPRKCA
SCHEMBL6976861 0.73 HTR6 (0.53) CYP1A2HTR6PRKD3PRKCGPRKCB
SCHEMBL840342 0.73 TDP1 (0.61) CYP1A2SMN1; SMN2LMNARAB9AALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0855391-B1 NOVEL ISOQUINOLINE DERIVATIVES DAIICHI SEIYAKU CO (JP) 2003-10-15 EP disclosed
US-5959107-A Isoquinoline derivatives SNOW BRAND MILK PRODUCTS CO., LTD. (JP) 1999-09-28 US disclosed
EP-0855391-A1 NOVEL ISOQUINOLINE DERIVATIVES SNOW BRAND MILK PRODUCTS CO., LTD. (JP) 1998-07-29 EP disclosed