SCHEMBL6967217

SCHEMBL6967217

COc1cccc(CBr)c1[N+](=O)[O-]

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 5/20 0.53
TDP1 Q9NUW8 3/20 0.53
L3MBTL1 Q9Y468 3/20 0.47
HPGD P15428 1/20 0.47
KDM4E B2RXH2 2/20 0.42
POLB P06746 1/20 0.42
CTDSP1 Q9GZU7 1/20 0.42
KMT2A Q03164 5/20 0.41
MEN1 O00255 4/20 0.41
NPC1 O15118 2/20 0.41
RAB9A P51151 2/20 0.41
SMN1; SMN2 Q16637 1/20 0.41
MAPT P10636 4/20 0.41
HTR1A P08908 1/20 0.40
ADRA1D P25100 1/20 0.40
ADRA1A P35348 1/20 0.40
ADRA1B P35368 1/20 0.40
GAA P10253 4/20 0.40
PKM P14618 2/20 0.40
MAPK1 P28482 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8217655 0.86 ALDH1A1 (0.52) ALDH1A1TDP1L3MBTL1HPGDKDM4E
SCHEMBL18138416 0.84 ALDH1A1 (0.50) ALDH1A1TDP1L3MBTL1HPGDKDM4E
SCHEMBL2027979 0.83 ALDH1A1 (0.46) ALDH1A1TDP1HPGDNPC1RAB9A
SCHEMBL16154026 0.83 HPGD (0.50) ALDH1A1TDP1L3MBTL1HPGDKDM4E
SCHEMBL194253 0.83 TDP1 (0.49) ALDH1A1TDP1L3MBTL1HPGDKDM4E
SCHEMBL8432682 0.83 ALDH1A1 (0.49) ALDH1A1TDP1L3MBTL1HPGDKDM4E
SCHEMBL27946152 0.83 ALDH1A1 (0.49) ALDH1A1TDP1L3MBTL1HPGDKDM4E
SCHEMBL13181024 0.81 ALDH1A1 (0.47) ALDH1A1TDP1L3MBTL1HPGDKDM4E
SCHEMBL1961457 0.81 TDP1 (0.63) ALDH1A1TDP1L3MBTL1HPGDKDM4E
SCHEMBL3779733 0.81 NPC1 (0.36) ALDH1A1TDP1HPGDPOLBKMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 9 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9499528-B2 Class of near infrared molecular probes for biological applications THE UNIVERSITY OF AKRON (US) 2016-11-22 US disclosed
US-20140303376-A1 CLASS OF NEAR INFRARED MOLECULAR PROBES FOR BIOLOGICAL APPLICATIONS THE UNIVERSITY OF AKRON 2014-10-09 US disclosed
EP-0955294-B1 Imidazolyl-alkenoic acid SMITHKLINE BEECHAM CORP (US) 2003-09-24 EP disclosed
EP-0955294-A2 Imidazolyl-alkenoic acid SMITHKLINE BEECHAM CORPORATION (US) 1999-11-10 EP disclosed
US-5418250-A Hypotensive SMITHKLINE BEECHAM CORPORATION (US) 1995-05-23 US disclosed
US-5312828-A Substituted imidazoles having angiotensin II receptor blocking activity SMITHKLINE BEECHAM CORPORATION A CORP. OF PENNSYLVANIA 1994-05-17 US disclosed
US-5185351-A Hypotensive agents; for treatment of congestive heart failure, renal failure and glaucoma SMITHKLINE BEECHAM CORPORATION (US) 1993-02-09 US disclosed
EP-0403158-A2 Imidazolyl-alkenoic acids SMITHKLINE BEECHAM CORPORATION (US) 1990-12-19 EP disclosed
EP-0403159-A2 Imidazolyl-alkenoic acids SMITHKLINE BEECHAM CORPORATION (US) 1990-12-19 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20140303376-A1 CLASS OF NEAR INFRARED MOLECULAR PROBES FOR BIOLOGICAL APPLICATIONS ZKSCAN2, ZRANB2, ZNF787 ALDH1A1 1141/4885TDP1 3397/4885L3MBTL1 2445/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.