Oxalic Acid

Oxalic Acid

SCHEMBL6967439

N=C(Nc1ccc(CNC(=O)OCc2ccccc2)cc1)c1cccs1.O=C(O)C(=O)O

nearest known ligand 0.52

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

OPRM1SLC6A4

The experimentally established mechanism targets of Oxalic Acid. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 1/20 0.49
RAB9A P51151 1/20 0.49
HPGD P15428 2/20 0.48
HDAC1 Q13547 3/20 0.48
PLAU P00749 1/20 0.47
NAMPT P43490 1/20 0.46
HDAC2 Q92769 2/20 0.46
HDAC3 O15379 1/20 0.46
L3MBTL1 Q9Y468 1/20 0.45
POLB P06746 1/20 0.44
MEN1 O00255 3/20 0.44
KMT2A Q03164 3/20 0.44
KDM4E B2RXH2 1/20 0.44
TSHR P16473 1/20 0.43
ALDH1A1 P00352 1/20 0.43
TP53 P04637 1/20 0.43
MMP2 P08253 1/20 0.43
MMP9 P14780 1/20 0.43
KDM1A O60341 2/20 0.42
MAOA P21397 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9037862 0.98 NPC1 (0.51) NPC1RAB9AHPGDHDAC1PLAU
SCHEMBL6968097 0.81 KDM4E (0.60) NPC1RAB9AHPGDHDAC1HDAC2
Oxalic Acid SCHEMBL6967537 0.80 MEN1 (0.44) NPC1RAB9AHPGDNAMPTL3MBTL1
SCHEMBL6968442 0.79 HPGD (0.59) NPC1RAB9AHPGDHDAC1L3MBTL1
SCHEMBL6963445 0.79 MEN1 (0.49) NPC1RAB9AHPGDL3MBTL1POLB
SCHEMBL10389709 0.79 POLB (0.64) NPC1RAB9AHDAC1PLAUNAMPT
SCHEMBL8148056 0.78 POLB (0.49) NPC1RAB9AHPGDL3MBTL1POLB
SCHEMBL6966981 0.77 HPGD (0.57) NPC1HPGDHDAC1HDAC2HDAC3
SCHEMBL9218989 0.77 MEN1 (0.45) NPC1RAB9AHPGDNAMPTL3MBTL1
SCHEMBL6958634 0.76 NPC1 (0.52) NPC1RAB9AMEN1KMT2AKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0713483-B1 AMIDINE DERIVATIVES WITH NITRIC OXIDE SYNTHETASE ACTIVITIES ASTRAZENECA AB (SE) 2003-01-15 EP disclosed
US-6030985-A Amidine derivatives with nitric oxide synthetase activities ASTRA AKTIEBOLAG (SE) 2000-02-29 US disclosed
US-5807885-A Amidine derivatives with nitric oxide synthetase activities ASTRA AKTIEBOLAG (SE) 1998-09-15 US disclosed
EP-0713483-A1 AMIDINE DERIVATIVES WITH NITRIC OXIDE SYNTHETASE ACTIVITIES Astra Aktiebolag (SE) 1996-05-29 EP disclosed
WO-1995005363-A1 AMIDINE DERIVATIVES WITH NITRIC OXIDE SYNTHETASE ACTIVITIES ASTRA AKTIEBOLAG (SE) 1995-02-23 WO disclosed