SCHEMBL6967716

SCHEMBL6967716

O=C(O)CC(NC(=O)COCc1ccccc1)c1ccccc1

nearest known ligand 0.52

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 4/20 0.49
POLB P06746 1/20 0.48
HTT P42858 2/20 0.48
ALDH1A1 P00352 1/20 0.48
NCOA1 Q15788 1/20 0.48
NCOA3 Q9Y6Q9 1/20 0.48
ITGB3 P05106 5/20 0.46
ITGA2B P08514 4/20 0.46
ITGAV P06756 2/20 0.46
ITGB5 P18084 2/20 0.46
ITGB6 P18564 1/20 0.46
CASP1 P29466 1/20 0.45
PTPRC P08575 1/20 0.45
PTPN1 P18031 1/20 0.45
TSHR P16473 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2249845 0.81 TSHR (0.67) SMN1; SMN2POLBHTTALDH1A1ITGB3
SCHEMBL6956276 0.80 CNR2 (0.65) SMN1; SMN2HTTALDH1A1NCOA1NCOA3
SCHEMBL28760324 0.80 CNR2 (0.65) SMN1; SMN2HTTALDH1A1NCOA1NCOA3
SCHEMBL27558113 0.80 CNR2 (0.65) SMN1; SMN2HTTALDH1A1NCOA1NCOA3
SCHEMBL6156731 0.79 CASP1 (0.60) ALDH1A1CASP1
SCHEMBL6955527 0.79 CASP1 (0.60) ALDH1A1CASP1
SCHEMBL6156740 0.79 CASP1 (0.60) ALDH1A1CASP1
SCHEMBL6957157 0.79 SMN1; SMN2 (0.61) SMN1; SMN2POLBALDH1A1
SCHEMBL6963806 0.79 ATM (0.51) SMN1; SMN2HTTPTPRCPTPN1TSHR
SCHEMBL7146807 0.79 CYP3A4 (0.54) SMN1; SMN2HTTALDH1A1CASP1TSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1021424-B1 THIADIAZOLE AMIDE MMP INHIBITORS UPJOHN CO (US) 2003-02-26 EP disclosed
US-5830869-A METALLOPROTEASE INHIBITOR PHARMACIA & UPJOHN COMPANY 1998-11-03 US disclosed