SCHEMBL6969556

SCHEMBL6969556

OC1(c2ccc3[nH]cc(CCC4CCCN4)c3c2)CCCCC1

nearest known ligand 0.61

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
SLC6A4 P31645 5/20 0.61
HTR6 P50406 11/20 0.44
HTR1D P28221 1/20 0.39
HTR2A P28223 1/20 0.38
DRD2 P14416 1/20 0.38
DRD4 P21917 1/20 0.38
DRD3 P35462 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6966131 0.91 SLC6A4 (0.58) SLC6A4HTR6HTR2ADRD2DRD4
SCHEMBL6967764 0.91 SLC6A4 (0.58) SLC6A4HTR6HTR1DHTR2A
SCHEMBL6968409 0.81 SLC6A4 (0.48) SLC6A4HTR6HTR1DDRD2DRD4
SCHEMBL8506913 0.78 SLC6A4 (0.70) SLC6A4HTR6HTR1DHTR2ADRD2
SCHEMBL6968677 0.78 SLC6A4 (0.70) SLC6A4HTR6HTR1DHTR2ADRD2
SCHEMBL6969558 0.77 MPO (0.60) HTR1DHTR2ADRD3
SCHEMBL6962932 0.77 SLC6A4 (0.66) SLC6A4HTR6HTR1D
SCHEMBL8506286 0.76 SLC6A4 (0.67) SLC6A4HTR6HTR1D
SCHEMBL6969543 0.76 SLC6A4 (0.64) SLC6A4HTR6HTR1DHTR2A
SCHEMBL8506945 0.75 SLC6A4 (0.66) SLC6A4HTR6HTR1D

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0944595-B1 5-CYCLO INDOLE COMPOUNDS AS 5-HT1D RECEPTOR LIGANDS NPS ALLELIX CORP (CA) 2003-10-01 EP claimed
EP-0944595-B1 5-CYCLO INDOLE COMPOUNDS AS 5-HT1D RECEPTOR LIGANDS NPS ALLELIX CORP (CA) 2003-10-01 EP disclosed
US-5998438-A SEROTONIN RECEPTOR ANTAGONIST; HEADACHE THERAPY ALLELIX BIOPHARMACEUTICALS, INC. (CA) 1999-12-07 US disclosed