SCHEMBL6969558

SCHEMBL6969558

OC1(c2ccc3[nH]cc(CCN4CCCC4)c3c2)CCCCC1

nearest known ligand 0.60

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
MPO P05164 3/20 0.60
HTR2A P28223 3/20 0.59
HTR1D P28221 10/20 0.58
HTR1B P28222 10/20 0.58
DRD3 P35462 1/20 0.49
BRD4 O60885 1/20 0.48
HTR7 P34969 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6967767 0.91 HTR1D (0.59) MPOHTR2AHTR1DHTR1BDRD3
SCHEMBL6966135 0.90 MPO (0.57) MPOHTR2AHTR1DHTR1BDRD3
SCHEMBL6967771 0.88 MPO (0.55) MPOHTR2AHTR1DHTR1BDRD3
SCHEMBL6968414 0.85 DRD3 (0.56) MPOHTR2AHTR1DHTR1BDRD3
SCHEMBL6970858 0.81 MPO (0.58) MPOHTR2AHTR1DHTR1BBRD4
SCHEMBL6968234 0.81 HTR1D (0.53) MPOHTR2AHTR1DHTR1BDRD3
SCHEMBL26989598 0.80 HTR7 (0.70) MPOHTR2AHTR1DHTR1BDRD3
SCHEMBL6968418 0.79 MPO (0.45) MPOHTR2AHTR1DHTR1BBRD4
SCHEMBL27095364 0.78 HTR7 (0.71) MPOHTR2AHTR1DHTR1BDRD3
SCHEMBL6969556 0.77 SLC6A4 (0.61) HTR2AHTR1DDRD3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0944595-B1 5-CYCLO INDOLE COMPOUNDS AS 5-HT1D RECEPTOR LIGANDS NPS ALLELIX CORP (CA) 2003-10-01 EP claimed
EP-0944595-B1 5-CYCLO INDOLE COMPOUNDS AS 5-HT1D RECEPTOR LIGANDS NPS ALLELIX CORP (CA) 2003-10-01 EP disclosed
US-5998438-A SEROTONIN RECEPTOR ANTAGONIST; HEADACHE THERAPY ALLELIX BIOPHARMACEUTICALS, INC. (CA) 1999-12-07 US disclosed