SCHEMBL6969691

SCHEMBL6969691

FC(F)(F)c1ccc(Cl)c(COCC2CCc3c(ncn3C(c3ccccc3)(c3ccccc3)c3ccccc3)C2)c1

nearest known ligand 0.33

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
DDR1 Q08345 1/20 0.33
NR1H2 P55055 1/20 0.33
FFAR4 Q5NUL3 2/20 0.33
SLC6A2 P23975 2/20 0.32
SLC6A4 P31645 2/20 0.32
FFAR1 O14842 1/20 0.31
DRD2 P14416 1/20 0.30
HTR2A P28223 1/20 0.30
HTR2C P28335 1/20 0.30
HTR2B P41595 1/20 0.30
SIGMAR1 Q99720 1/20 0.30
SCD O00767 1/20 0.30
TRAP1 Q12931 1/20 0.30
PTGDR2 Q9Y5Y4 1/20 0.30
P2RX7 Q99572 1/20 0.30
MRGPRX4 Q96LA9 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6969572 0.93 DDR1 (0.33) DDR1NR1H2FFAR4SLC6A2SLC6A4
SCHEMBL6958250 0.85 TACR1 (0.40) SLC6A4SIGMAR1
SCHEMBL6958774 0.85 TACR1 (0.36) DRD2HTR2AHTR2CHTR2BSIGMAR1
SCHEMBL6956374 0.84 P2RX7 (0.36) NR1H2FFAR4SLC6A2SLC6A4P2RX7
SCHEMBL6963452 0.80 CHRNB2 (0.43)
SCHEMBL7133170 0.80 CHRM1 (0.38) SLC6A2SLC6A4HTR2CHTR2BPTGDR2
SCHEMBL6957912 0.79 HTR2A (0.35) SLC6A4HTR2AHTR2CHTR2BSIGMAR1
SCHEMBL6966314 0.78 TACR1 (0.40) SIGMAR1
SCHEMBL6965989 0.78 CYP19A1 (0.32) FFAR4FFAR1
SCHEMBL6958015 0.78 TACR1 (0.36) DRD2HTR2AHTR2CHTR2BSIGMAR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6610721-B2 Imidazo heterocyclic compounds NOVO NORDISK A/S (DK) 2003-08-26 US disclosed
EP-1268483-A1 CONDENSED IMIDAZOLES AS HISTAMINE H3 RECEPTOR LIGANDS NOVO NORDISK A/S (DK) 2003-01-02 EP disclosed
US-20010049385-A1 Imidazo heterocyclic compounds HIGH POINT PHARMACEUTICALS, LLC 2001-12-06 US disclosed
WO-2001068651-A1 CONDENSED IMIDAZOLES AS HISTAMINE H3 RECEPTOR LIGANDS NOVO NORDISK A/S (DK) 2001-09-20 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20010049385-A1 Imidazo heterocyclic compounds HRH4, HRH3, HRH2 DDR1 4282/4885NR1H2 237/4885FFAR4 617/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.