SCHEMBL6970129

SCHEMBL6970129

CC(C)c1nc(CNC(N)=O)n(Cc2ccccn2)c1Sc1cccc(F)c1

nearest known ligand 0.40

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
S1PR3 Q99500 10/20 0.40
KMT2A Q03164 1/20 0.39
ADORA2A P29274 1/20 0.38
ADORA1 P30542 1/20 0.38
GRIN1 Q05586 2/20 0.37
GRIN2B Q13224 2/20 0.37
ALDH1A1 P00352 3/20 0.36
P2RX7 Q99572 1/20 0.36
NTRK1 P04629 2/20 0.35
MAPT P10636 1/20 0.35
HPGD P15428 1/20 0.35
RAB9A P51151 1/20 0.35
SMN1; SMN2 Q16637 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6970221 0.93 S1PR3 (0.41) S1PR3ALDH1A1NTRK1
SCHEMBL7084143 0.92 S1PR3 (0.41) S1PR3KMT2AADORA2AADORA1GRIN1
SCHEMBL7082911 0.90 ALDH1A1 (0.40) S1PR3KMT2AALDH1A1MAPTRAB9A
SCHEMBL7085418 0.90 POLB (0.38) S1PR3KMT2AADORA2AADORA1GRIN1
SCHEMBL6970143 0.88 GRIN1 (0.38) S1PR3KMT2AGRIN1GRIN2BALDH1A1
SCHEMBL7078713 0.87 S1PR3 (0.39) S1PR3KMT2AGRIN1GRIN2BRAB9A
SCHEMBL7078313 0.87 CYP1A2 (0.44) S1PR3KMT2AALDH1A1MAPT
SCHEMBL6967980 0.86 GRIN1 (0.39) S1PR3KMT2AGRIN1GRIN2BALDH1A1
SCHEMBL6972948 0.86 GRIN1 (0.39) S1PR3GRIN1GRIN2B
SCHEMBL6974276 0.86 GRIN1 (0.37) S1PR3KMT2AADORA2AADORA1GRIN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0786455-B1 IMIDAZOLE DERIVATIVE SHIONOGI & CO (JP) 2003-12-03 EP disclosed
US-6147097-A METHOD FOR TREATING AIDS SHIONOGI & CO., LTD. (JP) 2000-11-14 US disclosed
US-5910506-A IMIDAZOLE DERIVATIVES, E.G.5-(3,5-DICHLOROPHENYLTHIO)-1,2-DIMETHYL-4-ISOPROPYL-1H-IMIDAZOLE; VIRICIDES; AIDS; NONTOXIC SHIONOGI & CO., LTD. (JP) 1999-06-08 US disclosed
EP-0786455-A1 IMIDAZOLE DERIVATIVE SHIONOGI & CO., LTD. (JP) 1997-07-30 EP disclosed