SCHEMBL6972948

SCHEMBL6972948

CC(C)c1nc(CN)n(Cc2ccccn2)c1Sc1cccc(F)c1

nearest known ligand 0.39

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
GRIN1 Q05586 10/20 0.39
GRIN2B Q13224 10/20 0.39
S1PR3 Q99500 1/20 0.34
KDM4E B2RXH2 1/20 0.32
SLC6A9 P48067 3/20 0.32
ALOX5AP P20292 1/20 0.32
TLR9 Q9NR96 1/20 0.31
TLR8 Q9NR97 1/20 0.31
TLR7 Q9NYK1 1/20 0.31
NOX4 Q9NPH5 2/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6974115 0.92 GRIN1 (0.38) GRIN1GRIN2BS1PR3KDM4ETLR7
SCHEMBL7078209 0.92 S1PR3 (0.34) GRIN1GRIN2BS1PR3KDM4EALOX5AP
SCHEMBL6967980 0.90 GRIN1 (0.39) GRIN1GRIN2BS1PR3KDM4ESLC6A9
SCHEMBL6965115 0.89 TLR7 (0.36) GRIN1GRIN2BALOX5APTLR7
SCHEMBL6966820 0.89 GRIN1 (0.38) GRIN1GRIN2BS1PR3KDM4ESLC6A9
SCHEMBL6970143 0.89 GRIN1 (0.38) GRIN1GRIN2BS1PR3KDM4E
SCHEMBL6973313 0.89 GRIN1 (0.38) GRIN1GRIN2BS1PR3KDM4ESLC6A9
SCHEMBL6962202 0.88 GRM5 (0.38) GRIN1GRIN2BKDM4EALOX5APNOX4
SCHEMBL7078156 0.88 GRIN1 (0.36) GRIN1GRIN2BS1PR3
SCHEMBL6960568 0.88 GRIN1 (0.37) GRIN1GRIN2BS1PR3KDM4EALOX5AP

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0786455-B1 IMIDAZOLE DERIVATIVE SHIONOGI & CO (JP) 2003-12-03 EP disclosed
US-6147097-A METHOD FOR TREATING AIDS SHIONOGI & CO., LTD. (JP) 2000-11-14 US disclosed
EP-0786455-A1 IMIDAZOLE DERIVATIVE SHIONOGI & CO., LTD. (JP) 1997-07-30 EP disclosed