SCHEMBL6970485

SCHEMBL6970485

COc1ccc(COCc2nc(C(C)C)c(Sc3cccc([N+](=O)[O-])c3)n2C)cc1

nearest known ligand 0.42

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.42
MAPT P10636 6/20 0.39
MEN1 O00255 3/20 0.39
KMT2A Q03164 3/20 0.39
SMN1; SMN2 Q16637 2/20 0.39
CNR2 P34972 3/20 0.38
ACHE P22303 2/20 0.38
POLB P06746 1/20 0.37
NFE2L2 Q16236 1/20 0.36
CNR1 P21554 1/20 0.36
PKM P14618 1/20 0.36
MAOB P27338 1/20 0.36
ALOX5 P09917 1/20 0.36
GAA P10253 1/20 0.36
CYP3A4 P08684 1/20 0.36
CYP2C9 P11712 1/20 0.36
CYP2C19 P33261 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8801589 0.86 HSP90AA1 (0.38) ALDH1A1MAPTMEN1KMT2ASMN1; SMN2
SCHEMBL6966985 0.84 MAPT (0.35) ALDH1A1MAPTMEN1KMT2ASMN1; SMN2
SCHEMBL6970784 0.84 HSP90AA1 (0.36) ALDH1A1MAPTMEN1KMT2ASMN1; SMN2
SCHEMBL6960973 0.81 MAPT (0.39) ALDH1A1MAPTMEN1KMT2ASMN1; SMN2
SCHEMBL6960667 0.81 KMT2A (0.41) ALDH1A1MAPTMEN1KMT2ASMN1; SMN2
SCHEMBL6962522 0.81 CYP2C9 (0.40) ALDH1A1MAPTMEN1KMT2ASMN1; SMN2
SCHEMBL6969746 0.81 MEN1 (0.40) ALDH1A1MAPTMEN1KMT2ASMN1; SMN2
SCHEMBL7085473 0.81 MEN1 (0.35) ALDH1A1MAPTMEN1KMT2ASMN1; SMN2
SCHEMBL6973531 0.80 CNR2 (0.39) ALDH1A1MAPTMEN1KMT2ASMN1; SMN2
SCHEMBL6956933 0.80 HSP90AA1 (0.41) ALDH1A1MAPTKMT2ASMN1; SMN2ACHE

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0786455-B1 IMIDAZOLE DERIVATIVE SHIONOGI & CO (JP) 2003-12-03 EP claimed
EP-0786455-B1 IMIDAZOLE DERIVATIVE SHIONOGI & CO (JP) 2003-12-03 EP disclosed
US-6147097-A METHOD FOR TREATING AIDS SHIONOGI & CO., LTD. (JP) 2000-11-14 US disclosed
US-5910506-A IMIDAZOLE DERIVATIVES, E.G.5-(3,5-DICHLOROPHENYLTHIO)-1,2-DIMETHYL-4-ISOPROPYL-1H-IMIDAZOLE; VIRICIDES; AIDS; NONTOXIC SHIONOGI & CO., LTD. (JP) 1999-06-08 US disclosed
EP-0786455-A1 IMIDAZOLE DERIVATIVE SHIONOGI & CO., LTD. (JP) 1997-07-30 EP disclosed