SCHEMBL6973531

SCHEMBL6973531

COc1ccc(COCc2nc(C(C)C)c(Sc3cccc([N+](=O)[O-])c3)[nH]2)cc1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CNR2 P34972 1/20 0.39
KCNJ1 P48048 1/20 0.39
MAPT P10636 6/20 0.39
MEN1 O00255 4/20 0.39
KMT2A Q03164 4/20 0.39
ADORA2A P29274 1/20 0.38
NFE2L2 Q16236 1/20 0.38
ALDH1A1 P00352 3/20 0.37
PKM P14618 2/20 0.37
MAOB P27338 1/20 0.37
ALOX5 P09917 1/20 0.37
LMNA P02545 3/20 0.37
SMN1; SMN2 Q16637 3/20 0.36
L3MBTL1 Q9Y468 1/20 0.36
NPC1 O15118 1/20 0.36
GAA P10253 1/20 0.36
NFKB1 P19838 1/20 0.36
MAPK1 P28482 1/20 0.36
STAT1 P42224 1/20 0.36
HTT P42858 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6973717 0.84 LMNA (0.35) MAPTMEN1KMT2AALDH1A1LMNA
SCHEMBL5029294 0.81 DHFR (0.41) MEN1KMT2AALDH1A1MAOBLMNA
SCHEMBL6970485 0.80 ALDH1A1 (0.42) CNR2MAPTMEN1KMT2ANFE2L2
SCHEMBL6962307 0.79 CYP1A2 (0.35) ALDH1A1LMNASMN1; SMN2NPC1HTT
SCHEMBL14439826 0.76 TSHR (0.39) ALDH1A1ALOX5
SCHEMBL6964698 0.75 LMNA (0.36) LMNARAB9A
SCHEMBL14001841 0.74 DHFR (0.40) MAPTALDH1A1ALOX5SMN1; SMN2NPC1
SCHEMBL8801594 0.73 HSP90AA1 (0.39) MAPTMEN1KMT2AALDH1A1ALOX5
SCHEMBL6966442 0.73 HSP90AA1 (0.43) MAPTMEN1KMT2AALDH1A1ALOX5
SCHEMBL6975315 0.72 HSP90AA1 (0.39) MAPTMEN1KMT2AALDH1A1PKM

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0786455-B1 IMIDAZOLE DERIVATIVE SHIONOGI & CO (JP) 2003-12-03 EP disclosed
US-6147097-A METHOD FOR TREATING AIDS SHIONOGI & CO., LTD. (JP) 2000-11-14 US disclosed
US-5910506-A IMIDAZOLE DERIVATIVES, E.G.5-(3,5-DICHLOROPHENYLTHIO)-1,2-DIMETHYL-4-ISOPROPYL-1H-IMIDAZOLE; VIRICIDES; AIDS; NONTOXIC SHIONOGI & CO., LTD. (JP) 1999-06-08 US disclosed
EP-0786455-A1 IMIDAZOLE DERIVATIVE SHIONOGI & CO., LTD. (JP) 1997-07-30 EP disclosed