SCHEMBL6966985

SCHEMBL6966985

COc1ccc(COCc2nc(C(C)C)c(Sc3cccc(Cl)c3)n2C)cc1

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPT P10636 4/20 0.35
TP53 P04637 2/20 0.35
DHODH Q02127 1/20 0.35
LMNA P02545 1/20 0.34
KMT2A Q03164 4/20 0.33
ALDH1A1 P00352 2/20 0.33
DHFR P00374 2/20 0.33
PPP1CA P62136 1/20 0.33
KDM4E B2RXH2 1/20 0.33
HPGD P15428 1/20 0.33
POLB P06746 1/20 0.33
MEN1 O00255 2/20 0.33
NPSR1 Q6W5P4 1/20 0.33
TDP1 Q9NUW8 1/20 0.33
L3MBTL1 Q9Y468 1/20 0.33
CYP3A4 P08684 1/20 0.32
MAOB P27338 2/20 0.32
MAOA P21397 1/20 0.32
GAA P10253 1/20 0.32
SMN1; SMN2 Q16637 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6964520 0.91 DHODH (0.34) MAPTTP53DHODHALDH1A1DHFR
SCHEMBL6962017 0.90 TDP1 (0.39) MAPTTP53LMNAKMT2AALDH1A1
SCHEMBL6970485 0.84 ALDH1A1 (0.42) MAPTKMT2AALDH1A1POLBMEN1
SCHEMBL7078933 0.82 MAOB (0.35) MAPTTP53KMT2AALDH1A1PPP1CA
SCHEMBL6969238 0.82 VCP (0.38) DHODHKDM4ETDP1L3MBTL1SMN1; SMN2
SCHEMBL6974846 0.80 MEN1 (0.36) MAPTTP53DHODHKMT2ADHFR
SCHEMBL6965629 0.80 DHFR (0.33) MAPTTP53DHODHLMNAALDH1A1
SCHEMBL6974229 0.80 MAPT (0.34) MAPTTP53DHODHLMNAKMT2A
SCHEMBL14439857 0.79 DHODH (0.39) MAPTTP53DHODHALDH1A1HPGD
SCHEMBL6957630 0.79 DHODH (0.39) MAPTTP53DHODHALDH1A1HPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0786455-B1 IMIDAZOLE DERIVATIVE SHIONOGI & CO (JP) 2003-12-03 EP claimed
EP-0786455-B1 IMIDAZOLE DERIVATIVE SHIONOGI & CO (JP) 2003-12-03 EP disclosed
US-6147097-A METHOD FOR TREATING AIDS SHIONOGI & CO., LTD. (JP) 2000-11-14 US disclosed
US-5910506-A IMIDAZOLE DERIVATIVES, E.G.5-(3,5-DICHLOROPHENYLTHIO)-1,2-DIMETHYL-4-ISOPROPYL-1H-IMIDAZOLE; VIRICIDES; AIDS; NONTOXIC SHIONOGI & CO., LTD. (JP) 1999-06-08 US disclosed
EP-0786455-A1 IMIDAZOLE DERIVATIVE SHIONOGI & CO., LTD. (JP) 1997-07-30 EP disclosed