SCHEMBL6970659

SCHEMBL6970659

CN(C)CCc1cn(C(=O)c2ccccc2)c2ccc(C3C=COCC3)cc12

nearest known ligand 0.61

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
HTR6 P50406 11/20 0.61
HTR7 P34969 5/20 0.61
HTR1A P08908 3/20 0.61
HTR1D P28221 3/20 0.61
HTR1B P28222 3/20 0.61
HTR1F P30939 3/20 0.61
DRD2 P14416 2/20 0.35
DRD3 P35462 2/20 0.35
MTNR1A P48039 1/20 0.35
HTR1E P28566 1/20 0.35
BCHE P06276 1/20 0.35
AKR1C3 P42330 3/20 0.33
AKR1C4 P17516 1/20 0.33
PTGS1 P23219 1/20 0.33
AKR1C2 P52895 1/20 0.33
SCN9A Q15858 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6976877 0.80 HTR6 (0.61) HTR6HTR7HTR1AHTR1DHTR1B
SCHEMBL6976881 0.78 HTR6 (0.62) HTR6HTR7HTR1AHTR1DHTR1B
SCHEMBL8508379 0.77 HTR6 (0.61) HTR6HTR7HTR1AHTR1DHTR1B
SCHEMBL7443507 0.76 HTR6 (1.00) HTR6HTR7HTR1AHTR1DHTR1B
Acetic Acid SCHEMBL8508236 0.76 HTR6 (0.59) HTR6HTR7HTR1AHTR1DHTR1B
SCHEMBL6972524 0.75 HTR6 (0.77) HTR6HTR7HTR1AHTR1DHTR1B
SCHEMBL24877919 0.75 HTR6 (0.76) HTR6HTR7HTR1AHTR1DHTR1B
SCHEMBL30485872 0.75 HTR6 (0.76) HTR6HTR7HTR1AHTR1DHTR1B
SCHEMBL30485865 0.74 HTR6 (1.00) HTR6HTR7HTR1AHTR1DHTR1B
SCHEMBL5497004 0.74 HTR6 (1.00) HTR6HTR7HTR1AHTR1DHTR1B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0944595-B1 5-CYCLO INDOLE COMPOUNDS AS 5-HT1D RECEPTOR LIGANDS NPS ALLELIX CORP (CA) 2003-10-01 EP disclosed
US-5998438-A SEROTONIN RECEPTOR ANTAGONIST; HEADACHE THERAPY ALLELIX BIOPHARMACEUTICALS, INC. (CA) 1999-12-07 US disclosed