SCHEMBL6970868

SCHEMBL6970868

Cn1cc(CN2CCc3cc(N)ccc3C2)c2ccccc21

nearest known ligand 0.76

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.76
TSHR P16473 1/20 0.76
LMNA P02545 2/20 0.50
GLA P06280 1/20 0.50
HTR2A P28223 1/20 0.46
GPR84 Q9NQS5 1/20 0.43
DRD2 P14416 1/20 0.43
DRD4 P21917 1/20 0.43
DRD3 P35462 1/20 0.43
POLB P06746 1/20 0.42
HDAC8 Q9BY41 1/20 0.41
HDAC6 Q9UBN7 1/20 0.41
ABCB1 P08183 1/20 0.41
DHFR P00374 1/20 0.40
SMN1; SMN2 Q16637 1/20 0.40
MEN1 O00255 1/20 0.40
KMT2A Q03164 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6976524 0.78 DHFR (0.46) ALDH1A1TSHRLMNAGPR84DRD2
SCHEMBL6961921 0.76 POLB (0.55) ALDH1A1TSHRLMNAPOLBABCB1
SCHEMBL6974145 0.76 ALDH1A1 (0.43) ALDH1A1TSHRLMNADRD2DRD4
SCHEMBL6969248 0.75 BCHE (0.57) TSHRLMNAHTR2ADRD2DRD4
SCHEMBL6975713 0.75 ALDH1A1 (0.56) ALDH1A1TSHRLMNADRD2DRD4
SCHEMBL6964021 0.75 PDE4B (0.52) ALDH1A1TSHRDRD4POLBABCB1
SCHEMBL6392089 0.75 HTT (0.51) ALDH1A1TSHRLMNAHTR2ASMN1; SMN2
SCHEMBL6973388 0.74 TMEM97 (0.60) DRD2DRD4DRD3DHFRMEN1
SCHEMBL6960871 0.74 ALDH1A1 (0.40) ALDH1A1TSHRDRD2DRD4DRD3
SCHEMBL6974504 0.73 TP53 (0.57) ALDH1A1LMNASMN1; SMN2MEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0832069-B1 BIPHENYL-2-CARBOXYLIC ACID-TETRAHYDRO-ISOQUINOLIN-6-YL AMIDE DERIVATIVES, THEIR PREPARATION AND THEIR USE AS INHIBITORS OF MICROSOMAL TRIGLYCERIDE TRANSFER PROTEIN AND/OR APOLIPOPROTEIN B (Apo B) SECRETION PFIZER (US) 2003-03-05 EP disclosed
EP-1181954-A2 Biphenyl-2-carboxylic acid-tetrahydro-isoquinolin-6-yl amide derivatives, their preparation and use as inhibitors of microsomal triglyceride transfer protein and/or apolipoprotein B (ApoB) secretion PFIZER INC. (US) 2002-02-27 EP disclosed