SCHEMBL6971209

SCHEMBL6971209

CC(C)(C)[Si](C)(C)OCC1Cc2cc(N3C[C@H](CN)OC3=O)ccc2N1C(=O)OCc1ccccc1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GRM2 Q14416 6/20 0.35
PARP1 P09874 1/20 0.35
CETP P11597 1/20 0.35
MAOA P21397 2/20 0.34
HTR1A P08908 1/20 0.34
ADRA2A P08913 1/20 0.34
ADRA2B P18089 1/20 0.34
ADRA2C P18825 1/20 0.34
DRD1 P21728 1/20 0.34
HRH2 P25021 1/20 0.34
HTR1B P28222 1/20 0.34
HTR2A P28223 1/20 0.34
HTR2C P28335 1/20 0.34
HTR1E P28566 1/20 0.34
SLC6A4 P31645 1/20 0.34
HRH1 P35367 1/20 0.34
HTR2B P41595 1/20 0.34
TMEM97 Q5BJF2 1/20 0.34
SIGMAR1 Q99720 1/20 0.34
HRH3 Q9Y5N1 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6962353 0.93 MAOA (0.40) GRM2PARP1CETPMAOAHTR1A
SCHEMBL7081662 0.90 MAOA (0.46) MAOAMAOBLMNA
SCHEMBL7081661 0.90 MAOA (0.46) MAOAMAOBLMNA
SCHEMBL6972550 0.85 GRM2 (0.38) GRM2MAOAHTR1AADRA2AADRA2B
SCHEMBL6956015 0.78 MAOB (0.44) GRM2MAOAHTR1AADRA2AADRA2B
SCHEMBL6961334 0.78 GRM2 (0.40) GRM2CETPHTR1AADRA2AADRA2B
SCHEMBL6961781 0.77 SMN1; SMN2 (0.43) MAOAMAOBTP53TSHRALDH1A1
SCHEMBL27458038 0.77 MAOA (0.46) GRM2MAOAHTR1AADRA2AADRA2B
SCHEMBL6964490 0.77 MAOA (0.46) GRM2MAOAHTR1AADRA2AADRA2B
SCHEMBL7597985 0.76 GRM2 (0.38) GRM2MAOAHTR1AADRA2AADRA2B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1181288-B1 BICYCLIC OXAZOLIDINONES AS ANTIBACTERIAL AGENT UPJOHN CO (US) 2003-07-30 EP disclosed
US-20020143009-A1 Novel bicyclic oxazolidinones as antibacterial agents PHARMACIA & UPJOHN 2002-10-03 US disclosed
US-6387896-B1 GRAMNEGATIVE, GRAMPOSITVE BACTERIA PHARMACIA & UPJOHN CO. 2002-05-14 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20020143009-A1 Novel bicyclic oxazolidinones as antibacterial agents OXA1L, MRPL21, RPS4Y1 GRM2 4081/4885PARP1 1138/4885CETP 4549/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.