SCHEMBL6971574

SCHEMBL6971574

Cc1c(N(Cc2cccc(C#N)c2)C(=O)NC(C(=O)OCc2ccccc2)C(C)C)cnn1CC(C)C

nearest known ligand 0.38

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
IL1RN P18510 1/20 0.38
ERAP2 Q6P179 1/20 0.38
ERAP1 Q9NZ08 1/20 0.38
CTSB P07858 3/20 0.37
CTSK P43235 3/20 0.37
CTSL P07711 2/20 0.37
CTSS P25774 1/20 0.37
ADAMTS4 O75173 1/20 0.36
MMP13 P45452 1/20 0.36
ALDH1A1 P00352 1/20 0.36
MAPT P10636 1/20 0.36
PTGES O14684 7/20 0.36
NR3C1 P04150 1/20 0.36
MEN1 O00255 1/20 0.35
KMT2A Q03164 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6971488 0.90 ADAMTS4 (0.39) ADAMTS4MMP13ALDH1A1MAPTPTGES
SCHEMBL6964408 0.81 ALDH1A1 (0.43) ALDH1A1MAPTNR3C1
SCHEMBL6969060 0.80 ALDH1A1 (0.40) ALDH1A1MAPTPTGESNR3C1
SCHEMBL6973145 0.80 ALDH1A1 (0.40) ALDH1A1MAPTNR3C1
SCHEMBL6972441 0.80 ALDH1A1 (0.43) ADAMTS4MMP13ALDH1A1MAPTNR3C1
SCHEMBL6968547 0.79 ALDH1A1 (0.42) ALDH1A1MAPTNR3C1
SCHEMBL6973013 0.79 ALDH1A1 (0.40) ALDH1A1MAPTNR3C1
SCHEMBL6971108 0.78 ALDH1A1 (0.36) ALDH1A1MAPTPTGESNR3C1
SCHEMBL6971104 0.78 ALDH1A1 (0.36) ALDH1A1MAPTPTGESNR3C1
SCHEMBL6960549 0.76 MAPT (0.38) ALDH1A1MAPTNR3C1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1329160-A2 4-ACYLAMINOPYRAZOLE DERIVATIVES Sankyo Company, Limited (JP) 2003-07-23 EP disclosed