SCHEMBL6971599

SCHEMBL6971599

CC(C)c1nc(CN)n(Cc2ccncc2)c1Sc1cccc(F)c1

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GRIN1 Q05586 1/20 0.36
GRIN2B Q13224 1/20 0.36
ATM Q13315 2/20 0.33
KMT2A Q03164 1/20 0.33
LMNA P02545 1/20 0.33
TP53 P04637 1/20 0.33
KCNK13 Q9HB14 4/20 0.32
P2RX3 P56373 2/20 0.32
L3MBTL1 Q9Y468 1/20 0.32
CYP3A4 P08684 4/20 0.32
CYP17A1 P05093 1/20 0.32
CYP11B1 P15538 1/20 0.32
CYP11B2 P19099 1/20 0.32
TSHR P16473 1/20 0.32
HTT P42858 1/20 0.32
HTR1A P08908 1/20 0.31
DRD2 P14416 1/20 0.31
HTR2A P28223 1/20 0.31
HTR7 P34969 1/20 0.31
HTR6 P50406 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6975055 0.92 GRIN1 (0.35) GRIN1GRIN2BATMKMT2ALMNA
SCHEMBL7083358 0.91 KCNK13 (0.32) GRIN1GRIN2BKCNK13
SCHEMBL8109545 0.90 GRIN1 (0.36) GRIN1GRIN2BATMKMT2ALMNA
SCHEMBL6974887 0.89 GRIN1 (0.39) GRIN1GRIN2BATMCYP3A4CYP17A1
SCHEMBL6967360 0.89 IDO1 (0.36) KMT2AL3MBTL1HTTHTR1ADRD2
SCHEMBL6973510 0.88 GRIN1 (0.34) GRIN1GRIN2BATMKMT2ALMNA
SCHEMBL7086493 0.88 GRIN1 (0.35) GRIN1GRIN2BATMKMT2ALMNA
SCHEMBL6975612 0.88 GRIN1 (0.35) GRIN1GRIN2BATMKMT2ALMNA
SCHEMBL7082989 0.88 GRIN1 (0.35) GRIN1GRIN2BATMKMT2ALMNA
SCHEMBL7079161 0.87 GRIN1 (0.35) GRIN1GRIN2BATMKMT2ALMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0786455-B1 IMIDAZOLE DERIVATIVE SHIONOGI & CO (JP) 2003-12-03 EP disclosed
US-6147097-A METHOD FOR TREATING AIDS SHIONOGI & CO., LTD. (JP) 2000-11-14 US disclosed
US-5910506-A IMIDAZOLE DERIVATIVES, E.G.5-(3,5-DICHLOROPHENYLTHIO)-1,2-DIMETHYL-4-ISOPROPYL-1H-IMIDAZOLE; VIRICIDES; AIDS; NONTOXIC SHIONOGI & CO., LTD. (JP) 1999-06-08 US disclosed
EP-0786455-A1 IMIDAZOLE DERIVATIVE SHIONOGI & CO., LTD. (JP) 1997-07-30 EP disclosed