SCHEMBL6974887

SCHEMBL6974887

CC(C)c1nc(CN)n(Cc2cccnc2)c1Sc1cccc(F)c1

nearest known ligand 0.39

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
GRIN1 Q05586 13/20 0.39
GRIN2B Q13224 13/20 0.39
CYP11B2 P19099 1/20 0.34
TLR7 Q9NYK1 2/20 0.34
CYP3A4 P08684 2/20 0.34
CYP17A1 P05093 1/20 0.34
KDM4E B2RXH2 1/20 0.33
CYP1A2 P05177 1/20 0.33
CYP2D6 P10635 1/20 0.33
CYP2C19 P33261 1/20 0.33
ATM Q13315 1/20 0.33
ALDH1A1 P00352 1/20 0.33
POLB P06746 1/20 0.33
HPGD P15428 1/20 0.33
NPSR1 Q6W5P4 1/20 0.33
SRC P12931 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6972991 0.93 GRIN1 (0.38) GRIN1GRIN2BCYP11B2TLR7
SCHEMBL7084611 0.92 GRIN1 (0.39) GRIN1GRIN2BCYP11B2TLR7ALDH1A1
SCHEMBL7083464 0.90 GRIN1 (0.39) GRIN1GRIN2BCYP11B2CYP3A4CYP17A1
SCHEMBL6971599 0.89 GRIN1 (0.36) GRIN1GRIN2BCYP11B2CYP3A4CYP17A1
SCHEMBL6963828 0.89 GRIN1 (0.37) GRIN1GRIN2BCYP11B2TLR7CYP3A4
SCHEMBL6975548 0.89 GRIN1 (0.38) GRIN1GRIN2BCYP11B2CYP3A4CYP17A1
SCHEMBL7079895 0.89 GRIN1 (0.38) GRIN1GRIN2BCYP11B2TLR7CYP3A4
SCHEMBL6961326 0.89 GRIN1 (0.39) GRIN1GRIN2BCYP11B2ALDH1A1
SCHEMBL6965787 0.89 ALDH1A1 (0.38) GRIN1GRIN2BKDM4EALDH1A1HPGD
SCHEMBL6972848 0.88 TLR7 (0.38) TLR7CYP3A4KDM4ECYP2D6ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0786455-B1 IMIDAZOLE DERIVATIVE SHIONOGI & CO (JP) 2003-12-03 EP disclosed
US-6147097-A METHOD FOR TREATING AIDS SHIONOGI & CO., LTD. (JP) 2000-11-14 US disclosed
US-5910506-A IMIDAZOLE DERIVATIVES, E.G.5-(3,5-DICHLOROPHENYLTHIO)-1,2-DIMETHYL-4-ISOPROPYL-1H-IMIDAZOLE; VIRICIDES; AIDS; NONTOXIC SHIONOGI & CO., LTD. (JP) 1999-06-08 US disclosed
EP-0786455-A1 IMIDAZOLE DERIVATIVE SHIONOGI & CO., LTD. (JP) 1997-07-30 EP disclosed