SCHEMBL6967360

SCHEMBL6967360

CC(C)c1nc(CN)n(Cc2ccncc2)c1Sc1cccc(Cl)c1

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
IDO1 P14902 1/20 0.36
TDP1 Q9NUW8 3/20 0.35
ALDH1A1 P00352 3/20 0.34
MEN1 O00255 2/20 0.34
KMT2A Q03164 2/20 0.34
KDM4E B2RXH2 2/20 0.34
HPGD P15428 2/20 0.34
KCNH2 Q12809 1/20 0.33
POLB P06746 1/20 0.33
NPSR1 Q6W5P4 1/20 0.33
L3MBTL1 Q9Y468 1/20 0.33
PDE4D Q08499 1/20 0.33
NPC1 O15118 1/20 0.33
PDE4B Q07343 1/20 0.33
TYMS P04818 1/20 0.32
GRM5 P41594 2/20 0.32
HTR6 P50406 2/20 0.32
CCR2 P41597 1/20 0.32
CCR5 P51681 1/20 0.32
CSNK2A2 P19784 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6974232 0.92 IDO1 (0.35) IDO1TDP1ALDH1A1MEN1KMT2A
SCHEMBL6957548 0.90 KCNH2 (0.35) IDO1TDP1MEN1KMT2AKCNH2
SCHEMBL6965787 0.90 ALDH1A1 (0.38) IDO1TDP1ALDH1A1MEN1KMT2A
SCHEMBL7079909 0.90 IDO1 (0.36) IDO1TDP1ALDH1A1MEN1KMT2A
SCHEMBL6971599 0.89 GRIN1 (0.36) KMT2AKDM4EL3MBTL1HTR6HTR1A
SCHEMBL7084720 0.88 HTR3E (0.40) IDO1TDP1ALDH1A1MEN1KMT2A
SCHEMBL6972815 0.88 KDM4E (0.36) TDP1ALDH1A1KDM4EPIM1PIM3
SCHEMBL6972144 0.88 IDO1 (0.35) IDO1TDP1ALDH1A1MEN1KMT2A
SCHEMBL6959029 0.88 IDO1 (0.35) IDO1TDP1ALDH1A1MEN1KMT2A
SCHEMBL6963923 0.88 POLB (0.44) IDO1TDP1ALDH1A1MEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0786455-B1 IMIDAZOLE DERIVATIVE SHIONOGI & CO (JP) 2003-12-03 EP disclosed
US-6147097-A METHOD FOR TREATING AIDS SHIONOGI & CO., LTD. (JP) 2000-11-14 US disclosed
US-5910506-A IMIDAZOLE DERIVATIVES, E.G.5-(3,5-DICHLOROPHENYLTHIO)-1,2-DIMETHYL-4-ISOPROPYL-1H-IMIDAZOLE; VIRICIDES; AIDS; NONTOXIC SHIONOGI & CO., LTD. (JP) 1999-06-08 US disclosed
EP-0786455-A1 IMIDAZOLE DERIVATIVE SHIONOGI & CO., LTD. (JP) 1997-07-30 EP disclosed