SCHEMBL6972090

SCHEMBL6972090

Cc1ccc2nc(-c3cc(C(F)F)nn3-c3ccc(S(N)(=O)=O)cc3)sc2c1

nearest known ligand 0.66

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PTGS2 P35354 16/20 0.66
PTGS1 P23219 12/20 0.66
ABCB11 O95342 2/20 0.51
ALDH1A1 P00352 1/20 0.51
CCNE1 P24864 1/20 0.48
CDK2 P24941 1/20 0.48
CDK5 Q00535 1/20 0.48
CDK5R1 Q15078 1/20 0.48
PTGES O14684 2/20 0.45
PDPK1 O15530 2/20 0.45
HDAC3 O15379 1/20 0.45
CA12 O43570 1/20 0.45
PDE5A O76074 1/20 0.45
MT-CO2 P00403 1/20 0.45
CA1 P00915 1/20 0.45
CA2 P00918 1/20 0.45
LMNA P02545 1/20 0.45
CA3 P07451 1/20 0.45
CYP3A4 P08684 1/20 0.45
ALOX5 P09917 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6974226 0.91 PTGS2 (0.53) PTGS2PTGS1ALDH1A1CCNE1CDK2
SCHEMBL6982484 0.90 PTGS2 (0.56) PTGS2PTGS1ABCB11ALDH1A1CCNE1
SCHEMBL6978991 0.89 PTGS2 (0.64) PTGS2PTGS1ABCB11ALDH1A1CCNE1
SCHEMBL6973688 0.89 PTGS2 (0.66) PTGS2PTGS1ABCB11ALDH1A1CA12
SCHEMBL6972333 0.88 PTGS2 (0.64) PTGS2PTGS1ABCB11ALDH1A1CCNE1
SCHEMBL6978107 0.85 PTGS2 (0.65) PTGS2PTGS1ABCB11PTGESPDPK1
SCHEMBL6980897 0.84 PTGS2 (0.56) PTGS2PTGS1ABCB11ALDH1A1
SCHEMBL6974111 0.83 PTGS2 (0.54) PTGS2PTGS1ABCB11CCNE1CDK2
SCHEMBL6975857 0.82 PTGS2 (0.58) PTGS2PTGS1ABCB11ALDH1A1PTGES
SCHEMBL6972326 0.82 PTGS2 (0.48) PTGS2PTGS1ABCB11ALDH1A1CCNE1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1006114-B1 PYRAZOLE DERIVATIVES AND COX INHIBITORS CONTAINING THEM GRELAN PHARMACEUTICAL CO (JP) 2003-01-22 EP disclosed
US-6136831-A ANTIINFLAMMATORY AGENTS, GASTROINTESTINAL AGENTS, ENZYME INHIBITORS GRELAN PHARMACEUTICAL CO., LTD. (JP) 2000-10-24 US disclosed
EP-1006114-A1 PYRAZOLE DERIVATIVES AND COX INHIBITORS CONTAINING THEM Grelan Pharmaceutical Co., Ltd. (JP) 2000-06-07 EP disclosed