SCHEMBL6973688

SCHEMBL6973688

COc1ccc2nc(-c3cc(C(F)F)nn3-c3ccc(S(N)(=O)=O)cc3)sc2c1

nearest known ligand 0.66

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
PTGS2 P35354 16/20 0.66
PTGS1 P23219 11/20 0.66
ABCB11 O95342 1/20 0.55
ALDH1A1 P00352 1/20 0.55
CA1 P00915 3/20 0.46
CA2 P00918 3/20 0.46
CA9 Q16790 2/20 0.46
APP P05067 1/20 0.45
CA12 O43570 1/20 0.45
CA7 P43166 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6981308 0.92 PTGS1 (0.54) PTGS2PTGS1ABCB11ALDH1A1APP
SCHEMBL6972090 0.89 PTGS2 (0.66) PTGS2PTGS1ABCB11ALDH1A1CA1
SCHEMBL6982484 0.87 PTGS2 (0.56) PTGS2PTGS1ABCB11ALDH1A1
SCHEMBL6977030 0.86 PTGS2 (0.66) PTGS2PTGS1ABCB11CA1CA2
SCHEMBL6978991 0.86 PTGS2 (0.64) PTGS2PTGS1ABCB11ALDH1A1CA1
SCHEMBL6972333 0.84 PTGS2 (0.64) PTGS2PTGS1ABCB11ALDH1A1
SCHEMBL6980897 0.81 PTGS2 (0.56) PTGS2PTGS1ABCB11ALDH1A1
SCHEMBL6980721 0.81 PTGS2 (0.58) PTGS2PTGS1ABCB11ALDH1A1CA1
SCHEMBL213308 0.80 PTGS2 (1.00) PTGS2PTGS1ABCB11ALDH1A1CA1
SCHEMBL6352119 0.80 PTGS2 (1.00) PTGS2PTGS1ABCB11ALDH1A1CA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1006114-B1 PYRAZOLE DERIVATIVES AND COX INHIBITORS CONTAINING THEM GRELAN PHARMACEUTICAL CO (JP) 2003-01-22 EP disclosed
US-6136831-A ANTIINFLAMMATORY AGENTS, GASTROINTESTINAL AGENTS, ENZYME INHIBITORS GRELAN PHARMACEUTICAL CO., LTD. (JP) 2000-10-24 US disclosed
EP-1006114-A1 PYRAZOLE DERIVATIVES AND COX INHIBITORS CONTAINING THEM Grelan Pharmaceutical Co., Ltd. (JP) 2000-06-07 EP disclosed