SCHEMBL6972363

SCHEMBL6972363

Cc1cc(C)cc(N(c2cn[nH]c2)C(C#N)c2cccc(C#N)c2)c1

nearest known ligand 0.36

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
S1PR1 P21453 2/20 0.36
KCNA5 P22460 2/20 0.35
LRRK2 Q5S007 1/20 0.33
ROCK2 O75116 6/20 0.33
RPS6KB1 P23443 3/20 0.32
IDO1 P14902 1/20 0.32
ROCK1 Q13464 1/20 0.31
GRM5 P41594 1/20 0.30
CREBBP Q92793 1/20 0.30
MAOB P27338 1/20 0.30
FLT3 P36888 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6972370 0.66 S1PR1 (0.36) S1PR1KCNA5LRRK2
SCHEMBL28579957 0.64 ALDH1A1 (0.50) GRM5
SCHEMBL28971616 0.62 ALDH1A1 (0.52) S1PR1IDO1GRM5
SCHEMBL171405 0.62 IDO1 (0.59) LRRK2ROCK2IDO1MAOBFLT3
SCHEMBL29467167 0.61 HRH3 (0.55) ROCK2IDO1ROCK1
SCHEMBL22968664 0.61 HRH3 (0.55) ROCK2IDO1ROCK1
SCHEMBL28971594 0.61 S1PR1 (0.40) S1PR1KCNA5
Hydrochloric Acid SCHEMBL29271375 0.60 HRH3 (0.54) ROCK2IDO1ROCK1
Hydrochloric Acid SCHEMBL30986706 0.60 HRH3 (0.54) ROCK2IDO1ROCK1
SCHEMBL22435570 0.60 GLA (0.44) S1PR1CREBBP

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1329160-A2 4-ACYLAMINOPYRAZOLE DERIVATIVES Sankyo Company, Limited (JP) 2003-07-23 EP disclosed