SCHEMBL6972370

SCHEMBL6972370

Cc1n[nH]c(C)c1N(c1ccccc1)C(C#N)c1cccc(C#N)c1

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
S1PR1 P21453 2/20 0.36
LRRK2 Q5S007 1/20 0.33
EP300 Q09472 2/20 0.33
KCNN4 O15554 1/20 0.32
KCNA5 P22460 1/20 0.32
PIN1 Q13526 1/20 0.32
PLK1 P53350 1/20 0.32
SLC6A2 P23975 2/20 0.32
SLC6A4 P31645 2/20 0.32
MAPK1 P28482 1/20 0.32
ALDH1A1 P00352 2/20 0.32
HTT P42858 2/20 0.32
LMNA P02545 1/20 0.32
TSHR P16473 1/20 0.32
CRHBP P24387 1/20 0.32
CRHR2 Q13324 1/20 0.32
SMN1; SMN2 Q16637 1/20 0.32
NPSR1 Q6W5P4 1/20 0.32
CHEK1 O14757 1/20 0.31
AKT2 P31751 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6972138 0.71 LRRK2 (0.39) LRRK2EP300PIN1PLK1SLC6A2
SCHEMBL6972363 0.66 S1PR1 (0.36) S1PR1LRRK2KCNA5
SCHEMBL6966470 0.66 MEP1A (0.44) PIN1SLC6A2SLC6A4LMNA
SCHEMBL13367360 0.64 KCNA5 (0.46) S1PR1KCNN4KCNA5ALDH1A1HTT
SCHEMBL7093358 0.64 LMNA (0.50) ALDH1A1LMNATSHRSMN1; SMN2
SCHEMBL6971350 0.64 MEP1A (0.44) PIN1SLC6A2SLC6A4
SCHEMBL7095374 0.63 IDO1 (0.42) ALDH1A1LMNATSHRSMN1; SMN2
SCHEMBL17069276 0.63 TSHR (0.45) S1PR1SLC6A2SLC6A4ALDH1A1TSHR
SCHEMBL17069277 0.62 TSHR (0.48) S1PR1SLC6A2SLC6A4ALDH1A1TSHR
SCHEMBL11601064 0.62 TSHR (0.48) SLC6A2SLC6A4ALDH1A1HTTLMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1329160-A2 4-ACYLAMINOPYRAZOLE DERIVATIVES Sankyo Company, Limited (JP) 2003-07-23 EP disclosed