SCHEMBL6972447

SCHEMBL6972447

CC(C)c1c(Sc2ccccc2)nc(COCCO)n1Cc1ccncc1

nearest known ligand 0.33

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
MAPT P10636 2/20 0.33
TP53 P04637 1/20 0.33
TLR7 Q9NYK1 1/20 0.32
GSK3B P49841 1/20 0.32
KDM4E B2RXH2 1/20 0.32
CYP1A2 P05177 1/20 0.32
CYP3A4 P08684 1/20 0.32
CYP2D6 P10635 1/20 0.32
CYP2C9 P11712 1/20 0.32
CYP2C19 P33261 1/20 0.32
HIF1A Q16665 1/20 0.32
ALOX5AP P20292 1/20 0.31
S1PR3 Q99500 1/20 0.31
ALDH1A1 P00352 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7080472 0.90 CSNK2A2 (0.34) MAPTGSK3BKDM4ECYP1A2CYP3A4
SCHEMBL7086504 0.89 GRIN1 (0.33) TP53S1PR3
SCHEMBL6974063 0.88 KCNH2 (0.32)
SCHEMBL6967184 0.87 ENPP2 (0.31)
SCHEMBL6973406 0.86 KDM4E (0.36) MAPTTLR7GSK3BKDM4ECYP1A2
SCHEMBL6961316 0.86 PDE4A (0.36) MAPTCYP2D6CYP2C9CYP2C19ALDH1A1
SCHEMBL6961644 0.85 ACSS2 (0.34) ALDH1A1
SCHEMBL6967059 0.84 MAPT (0.33) MAPTTP53TLR7GSK3BKDM4E
SCHEMBL7079123 0.84 MEN1 (0.37) MAPTTP53KDM4ECYP1A2CYP2C9
SCHEMBL6973086 0.83 PIM1 (0.36) MAPTTP53TLR7KDM4ES1PR3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0786455-B1 IMIDAZOLE DERIVATIVE SHIONOGI & CO (JP) 2003-12-03 EP disclosed
US-6147097-A METHOD FOR TREATING AIDS SHIONOGI & CO., LTD. (JP) 2000-11-14 US disclosed
US-5910506-A IMIDAZOLE DERIVATIVES, E.G.5-(3,5-DICHLOROPHENYLTHIO)-1,2-DIMETHYL-4-ISOPROPYL-1H-IMIDAZOLE; VIRICIDES; AIDS; NONTOXIC SHIONOGI & CO., LTD. (JP) 1999-06-08 US disclosed
EP-0786455-A1 IMIDAZOLE DERIVATIVE SHIONOGI & CO., LTD. (JP) 1997-07-30 EP disclosed