SCHEMBL6972509

SCHEMBL6972509

CC(C)(CN1CCC(C#N)(NC(=O)CCC2CCCCC2)C1)c1ccccc1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CTSS P25774 10/20 0.46
CTSB P07858 2/20 0.41
CTSL P07711 1/20 0.41
OPRM1 P35372 2/20 0.41
OPRL1 P41146 2/20 0.41
KDM1A O60341 1/20 0.38
MAOB P27338 1/20 0.38
ALDH1A1 P00352 4/20 0.38
MEN1 O00255 1/20 0.38
KMT2A Q03164 1/20 0.38
TDP1 Q9NUW8 1/20 0.38
NPC1 O15118 1/20 0.38
HPGD P15428 1/20 0.38
NFKB1 P19838 1/20 0.38
RAB9A P51151 1/20 0.38
NFKB2 Q00653 1/20 0.38
RELA Q04206 1/20 0.38
SMN1; SMN2 Q16637 1/20 0.38
HSD17B10 Q99714 1/20 0.38
TP53 P04637 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6972505 0.86 CTSS (0.46) CTSSCTSBCTSLOPRM1OPRL1
SCHEMBL6972946 0.85 CTSS (0.59) CTSSCTSBCTSLOPRM1OPRL1
SCHEMBL5357132 0.84 CTSS (0.53) CTSSCTSL
SCHEMBL6965443 0.80 CTSS (0.54) CTSSCTSBCTSLALDH1A1HPGD
SCHEMBL5756837 0.78 CTSS (0.78) CTSS
SCHEMBL5756463 0.78 CTSS (0.78) CTSS
SCHEMBL14383653 0.78 CTSS (0.64) CTSSCTSBCTSL
SCHEMBL5357125 0.77 CTSS (0.44) CTSSCTSBCTSLOPRM1OPRL1
SCHEMBL6063791 0.77 CTSL (0.51) CTSSCTSBCTSLALDH1A1HPGD
SCHEMBL6836051 0.74 CTSL (0.53) CTSSCTSBCTSLALDH1A1NPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1218372-B1 NOVEL HETEROCYCLIC COMPOUNDS USEFUL AS REVERSIBLE INHIBITORS OF CYSTEINE PROTEASES BOEHRINGER INGELHEIM PHARMA (US) 2003-07-02 EP disclosed