SCHEMBL6972789

SCHEMBL6972789

CNCc1nc(C(C)C)c(Sc2ccccc2)n1Cc1ccccn1

nearest known ligand 0.35

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HRH3 Q9Y5N1 1/20 0.35
ALDH1A1 P00352 5/20 0.34
LMNA P02545 1/20 0.34
TAAR1 Q96RJ0 1/20 0.34
ALOX15 P16050 1/20 0.34
CYP1A2 P05177 2/20 0.34
CYP2C19 P33261 1/20 0.34
ALOX5AP P20292 1/20 0.34
TLR7 Q9NYK1 3/20 0.33
PIP4K2C Q8TBX8 2/20 0.32
MAPT P10636 2/20 0.32
CYP2D6 P10635 1/20 0.32
TSHR P16473 1/20 0.32
SMN1; SMN2 Q16637 1/20 0.32
TP53 P04637 1/20 0.32
MAOA P21397 1/20 0.32
MAOB P27338 1/20 0.32
KDM4E B2RXH2 1/20 0.32
NPSR1 Q6W5P4 1/20 0.32
KCNH2 Q12809 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6961462 0.89 GRIN1 (0.37) ALDH1A1CYP1A2CYP2C19MAPTTP53
SCHEMBL6970143 0.89 GRIN1 (0.38) ALDH1A1MAPTSMN1; SMN2KDM4E
SCHEMBL6974447 0.89 MEN1 (0.34) HRH3ALDH1A1ALOX5APTLR7MAPT
SCHEMBL6960222 0.89 S1PR3 (0.36) HRH3TLR7
SCHEMBL6965884 0.88 ALDH1A1 (0.41) ALDH1A1CYP1A2MAPTCYP2D6TSHR
SCHEMBL7082911 0.87 ALDH1A1 (0.40) ALDH1A1CYP1A2MAPTCYP2D6TSHR
SCHEMBL7077261 0.87 POLB (0.35) ALDH1A1LMNATLR7
SCHEMBL6965115 0.87 TLR7 (0.36) ALDH1A1LMNACYP1A2CYP2C19ALOX5AP
SCHEMBL6963974 0.87 ALDH1A1 (0.37) ALDH1A1LMNACYP1A2CYP2C19ALOX5AP
SCHEMBL7086006 0.86 ALOX5AP (0.33) ALDH1A1LMNACYP1A2CYP2C19ALOX5AP

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0786455-B1 IMIDAZOLE DERIVATIVE SHIONOGI & CO (JP) 2003-12-03 EP disclosed
US-6147097-A METHOD FOR TREATING AIDS SHIONOGI & CO., LTD. (JP) 2000-11-14 US disclosed
US-5910506-A IMIDAZOLE DERIVATIVES, E.G.5-(3,5-DICHLOROPHENYLTHIO)-1,2-DIMETHYL-4-ISOPROPYL-1H-IMIDAZOLE; VIRICIDES; AIDS; NONTOXIC SHIONOGI & CO., LTD. (JP) 1999-06-08 US disclosed
EP-0786455-A1 IMIDAZOLE DERIVATIVE SHIONOGI & CO., LTD. (JP) 1997-07-30 EP disclosed