SCHEMBL6972884

SCHEMBL6972884

CC(C)c1nc(COC(N)=O)n(C)c1Sc1cc(F)cc(F)c1

nearest known ligand 0.36

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
LMNA P02545 1/20 0.36
CYP1A2 P05177 1/20 0.32
CYP3A4 P08684 1/20 0.32
CYP2C9 P11712 1/20 0.32
CYP2C19 P33261 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6969319 0.91
SCHEMBL6973457 0.90 CYP1A2 (0.36) CYP1A2CYP3A4CYP2C9CYP2C19
SCHEMBL6969795 0.89 EPHX1 (0.37) LMNACYP1A2CYP3A4CYP2C9CYP2C19
SCHEMBL6972480 0.89
SCHEMBL6961197 0.88 LMNA (0.31) LMNA
SCHEMBL6973251 0.88 LMNA (0.36) LMNA
SCHEMBL6967644 0.87 GLA (0.32) LMNACYP1A2CYP3A4CYP2C9CYP2C19
SCHEMBL6972317 0.87 LMNA (0.32) LMNA
SCHEMBL6969451 0.87 MEN1 (0.38) LMNACYP1A2CYP3A4CYP2C9CYP2C19
SCHEMBL7083502 0.87 KDM4E (0.33)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0786455-B1 IMIDAZOLE DERIVATIVE SHIONOGI & CO (JP) 2003-12-03 EP disclosed
US-6147097-A METHOD FOR TREATING AIDS SHIONOGI & CO., LTD. (JP) 2000-11-14 US disclosed
US-5910506-A IMIDAZOLE DERIVATIVES, E.G.5-(3,5-DICHLOROPHENYLTHIO)-1,2-DIMETHYL-4-ISOPROPYL-1H-IMIDAZOLE; VIRICIDES; AIDS; NONTOXIC SHIONOGI & CO., LTD. (JP) 1999-06-08 US disclosed
EP-0786455-A1 IMIDAZOLE DERIVATIVE SHIONOGI & CO., LTD. (JP) 1997-07-30 EP disclosed