SCHEMBL6969795

SCHEMBL6969795

CC(C)c1nc(COC(N)=O)n(C)c1Sc1cccc(F)c1

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
EPHX1 P07099 2/20 0.37
MAOA P21397 2/20 0.35
MAOB P27338 2/20 0.35
SLC6A9 P48067 5/20 0.35
LMNA P02545 2/20 0.33
NOTUM Q6P988 1/20 0.33
PPARG P37231 1/20 0.33
MAPT P10636 1/20 0.33
CA2 P00918 1/20 0.33
CA4 P22748 1/20 0.33
ALDH1A1 P00352 1/20 0.32
L3MBTL1 Q9Y468 1/20 0.32
TP53 P04637 1/20 0.32
CYP1A2 P05177 2/20 0.32
CYP3A4 P08684 2/20 0.32
CYP2C9 P11712 2/20 0.32
CYP2C19 P33261 2/20 0.32
GAA P10253 1/20 0.32
CYP2D6 P10635 1/20 0.32
NPSR1 Q6W5P4 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7087401 0.91 EPHX1 (0.34) EPHX1MAOAMAOBSLC6A9LMNA
SCHEMBL6962728 0.91 CYP1A2 (0.40) EPHX1MAOAMAOBSLC6A9LMNA
SCHEMBL6965977 0.90 EPHX1 (0.35) EPHX1MAOAMAOBSLC6A9LMNA
SCHEMBL6972884 0.89 LMNA (0.36) LMNACYP1A2CYP3A4CYP2C9CYP2C19
SCHEMBL7084556 0.88 EPHX1 (0.34) EPHX1MAOAMAOBSLC6A9LMNA
SCHEMBL6969410 0.88 TOP2A (0.35) EPHX1MAOAMAOBSLC6A9LMNA
SCHEMBL6974432 0.88 EPHX1 (0.35) EPHX1MAOAMAOBSLC6A9LMNA
SCHEMBL6967291 0.88 ALOX12 (0.36) MAOAMAOBSLC6A9LMNANOTUM
SCHEMBL6969941 0.87 CYP1A2 (0.39) EPHX1LMNAMAPTL3MBTL1TP53
SCHEMBL6973934 0.84 EPHX1 (0.37) EPHX1MAOAMAOBSLC6A9LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0786455-B1 IMIDAZOLE DERIVATIVE SHIONOGI & CO (JP) 2003-12-03 EP disclosed
US-6147097-A METHOD FOR TREATING AIDS SHIONOGI & CO., LTD. (JP) 2000-11-14 US disclosed
US-5910506-A IMIDAZOLE DERIVATIVES, E.G.5-(3,5-DICHLOROPHENYLTHIO)-1,2-DIMETHYL-4-ISOPROPYL-1H-IMIDAZOLE; VIRICIDES; AIDS; NONTOXIC SHIONOGI & CO., LTD. (JP) 1999-06-08 US disclosed
EP-0786455-A1 IMIDAZOLE DERIVATIVE SHIONOGI & CO., LTD. (JP) 1997-07-30 EP disclosed