SCHEMBL6973313

SCHEMBL6973313

CC(C)c1nc(CCO)n(Cc2ccccn2)c1Sc1cccc(F)c1

nearest known ligand 0.38

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
GRIN1 Q05586 8/20 0.38
GRIN2B Q13224 8/20 0.38
S1PR3 Q99500 2/20 0.35
KDM4E B2RXH2 1/20 0.33
HRH1 P35367 1/20 0.33
KMT2A Q03164 1/20 0.32
ALDH1A1 P00352 1/20 0.32
MAPT P10636 1/20 0.32
HPGD P15428 1/20 0.32
RAB9A P51151 1/20 0.32
SMN1; SMN2 Q16637 1/20 0.32
TLR7 Q9NYK1 1/20 0.32
GCGR P47871 1/20 0.32
SLC6A9 P48067 2/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6974995 0.94 GRIN1 (0.36) GRIN1GRIN2BS1PR3KDM4EHRH1
SCHEMBL6967980 0.92 GRIN1 (0.39) GRIN1GRIN2BS1PR3KDM4EKMT2A
SCHEMBL6967358 0.92 S1PR3 (0.35) GRIN1GRIN2BS1PR3KDM4EHRH1
SCHEMBL6974115 0.91 GRIN1 (0.38) GRIN1GRIN2BS1PR3KDM4EHRH1
SCHEMBL6974453 0.89 ENPP2 (0.38) GRIN1GRIN2BS1PR3KMT2ASLC6A9
SCHEMBL7084157 0.89 TLR7 (0.37) KDM4EHRH1ALDH1A1RAB9ASMN1; SMN2
SCHEMBL7082472 0.89 ALDH1A1 (0.37) GRIN1GRIN2BKDM4EHRH1KMT2A
SCHEMBL6972948 0.89 GRIN1 (0.39) GRIN1GRIN2BS1PR3KDM4ETLR7
SCHEMBL6974365 0.88 GRIN1 (0.35) GRIN1GRIN2BS1PR3HRH1SLC6A9
SCHEMBL6974113 0.87 S1PR3 (0.38) GRIN1GRIN2BS1PR3KMT2ASLC6A9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0786455-B1 IMIDAZOLE DERIVATIVE SHIONOGI & CO (JP) 2003-12-03 EP disclosed
US-6147097-A METHOD FOR TREATING AIDS SHIONOGI & CO., LTD. (JP) 2000-11-14 US disclosed
US-5910506-A IMIDAZOLE DERIVATIVES, E.G.5-(3,5-DICHLOROPHENYLTHIO)-1,2-DIMETHYL-4-ISOPROPYL-1H-IMIDAZOLE; VIRICIDES; AIDS; NONTOXIC SHIONOGI & CO., LTD. (JP) 1999-06-08 US disclosed
EP-0786455-A1 IMIDAZOLE DERIVATIVE SHIONOGI & CO., LTD. (JP) 1997-07-30 EP disclosed