SCHEMBL6974115

SCHEMBL6974115

CC(C)c1nc(CCN)n(Cc2ccccn2)c1Sc1cccc(F)c1

nearest known ligand 0.38

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
GRIN1 Q05586 13/20 0.38
GRIN2B Q13224 13/20 0.38
HRH1 P35367 1/20 0.34
TLR7 Q9NYK1 1/20 0.33
KDM4E B2RXH2 1/20 0.33
S1PR3 Q99500 1/20 0.33
GNRHR P30968 2/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6969106 0.92 HRH1 (0.36) GRIN1GRIN2BHRH1TLR7S1PR3
SCHEMBL6972948 0.92 GRIN1 (0.39) GRIN1GRIN2BTLR7KDM4ES1PR3
SCHEMBL6973313 0.91 GRIN1 (0.38) GRIN1GRIN2BHRH1TLR7KDM4E
SCHEMBL6973209 0.89 HRH1 (0.40) GRIN1GRIN2BHRH1TLR7GNRHR
SCHEMBL6974995 0.89 GRIN1 (0.36) GRIN1GRIN2BHRH1TLR7KDM4E
SCHEMBL6967528 0.89 GRM5 (0.36) GRIN1GRIN2BHRH1TLR7KDM4E
SCHEMBL6967980 0.89 GRIN1 (0.39) GRIN1GRIN2BKDM4ES1PR3
SCHEMBL6974453 0.87 ENPP2 (0.38) GRIN1GRIN2BS1PR3
SCHEMBL6970143 0.87 GRIN1 (0.38) GRIN1GRIN2BKDM4ES1PR3
SCHEMBL6966820 0.87 GRIN1 (0.38) GRIN1GRIN2BKDM4ES1PR3GNRHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0786455-B1 IMIDAZOLE DERIVATIVE SHIONOGI & CO (JP) 2003-12-03 EP disclosed
US-6147097-A METHOD FOR TREATING AIDS SHIONOGI & CO., LTD. (JP) 2000-11-14 US disclosed
US-5910506-A IMIDAZOLE DERIVATIVES, E.G.5-(3,5-DICHLOROPHENYLTHIO)-1,2-DIMETHYL-4-ISOPROPYL-1H-IMIDAZOLE; VIRICIDES; AIDS; NONTOXIC SHIONOGI & CO., LTD. (JP) 1999-06-08 US disclosed
EP-0786455-A1 IMIDAZOLE DERIVATIVE SHIONOGI & CO., LTD. (JP) 1997-07-30 EP disclosed