SCHEMBL6973108

SCHEMBL6973108

CSc1ccc(-n2nc(C(F)(F)F)cc2-c2nc3ccccc3s2)cc1

nearest known ligand 0.51

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
PTGS2 P35354 11/20 0.51
PTGS1 P23219 9/20 0.51
NPSR1 Q6W5P4 1/20 0.41
MAPT P10636 1/20 0.40
RXFP1 Q9HBX9 1/20 0.40
P2RY6 Q15077 2/20 0.40
F2RL3 Q96RI0 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6978354 0.87 PTGS2 (0.49) PTGS2PTGS1F2RL3
SCHEMBL6976230 0.87 PTGS2 (0.49) PTGS2PTGS1F2RL3
SCHEMBL6976132 0.84 PTGS2 (0.48) PTGS2PTGS1
SCHEMBL6978032 0.84 PTGS2 (0.64) PTGS2PTGS1
SCHEMBL6976876 0.82 PTGS2 (0.64) PTGS2PTGS1
SCHEMBL6973119 0.76 P2RY6 (0.40) PTGS2PTGS1NPSR1MAPTP2RY6
SCHEMBL4032238 0.75 PTGS1 (0.74) PTGS2PTGS1NPSR1MAPT
SCHEMBL6973228 0.72 PTGS2 (0.64) PTGS2PTGS1
SCHEMBL25150243 0.72 PTGS2 (0.72) PTGS2PTGS1
SCHEMBL9273738 0.72 PTGS2 (0.72) PTGS2PTGS1NPSR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1006114-B1 PYRAZOLE DERIVATIVES AND COX INHIBITORS CONTAINING THEM GRELAN PHARMACEUTICAL CO (JP) 2003-01-22 EP disclosed
US-6136831-A ANTIINFLAMMATORY AGENTS, GASTROINTESTINAL AGENTS, ENZYME INHIBITORS GRELAN PHARMACEUTICAL CO., LTD. (JP) 2000-10-24 US disclosed
EP-1006114-A1 PYRAZOLE DERIVATIVES AND COX INHIBITORS CONTAINING THEM Grelan Pharmaceutical Co., Ltd. (JP) 2000-06-07 EP disclosed